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5SJP

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH N1(CCC1)C(=O)c2c(n(nc2)C)C(=O)Nc3cc(nc(c3)C)NC(NC(OCC)=O)=S, micromolar IC50=0.402697

Resources
File formatFile name (file size)
PDBx/mmCIF5sjp.cif.gz Display(275.84 KB)
5sjp.cif
PDBx/mmJSONall5sjp.json.gz Display (Tree)(170.31 KB)
5sjp.json
no-atom5sjp-noatom.json.gz Display (Header)(20.69 KB)
5sjp-noatom.json
add only5sjp-plus.json.gz Display(1015.00 B)
5sjp-plus.json
PDBMLall5sjp.xml.gz Display(377.43 KB)
5sjp.xml
no-atom5sjp-noatom.xml.gz Display(55.68 KB)
5sjp-noatom.xml
ext-atom5sjp-extatom.xml.gz Display(243.17 KB)
5sjp-extatom.xml
pdb_nextgenallpdb_00005sjp_xyz-enrich.cif.gz Display(301.09 KB)
pdb_00005sjp_xyz-enrich.cif
no-atompdb_00005sjp_xyz-no-atom-enrich.xml.gz Display(68.84 KB)
pdb_00005sjp_xyz-no-atom-enrich.xml
ng-only5sjp-plus.json.gz Display(3.42 KB)
5sjp-plus.json
PDBpdb5sjp.ent.gz Display(222.40 KB)
pdb5sjp.ent
RDF5sjp.rdf.gz Visualize(151.00 KB)
5sjp.rdf
Structure factorsr5sjpsf.ent.gz Display(9.01 MB)
r5sjpsf.ent
Biological unit (mmCIF format)5sjp-assembly1.cif.gz Display(71.75 KB)
5sjp-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5sjp-assembly2.cif.gz Display(71.86 KB)
5sjp-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

5sjp-assembly3.cif.gz Display(72.31 KB)
5sjp-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

5sjp-assembly4.cif.gz Display(68.97 KB)
5sjp-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5sjp.pdb1.gz Display(56.89 KB)
5sjp.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5sjp.pdb2.gz Display(56.98 KB)
5sjp.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

5sjp.pdb3.gz Display(57.45 KB)
5sjp.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

5sjp.pdb4.gz Display(54.89 KB)
5sjp.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5sjp_validation.pdf.gz Display(1.47 MB)
5sjp_validation.pdf
PDF-full5sjp_full_validation.pdf.gz Display(1.50 MB)
5sjp_full_validation.pdf
mmCIF5sjp_validation.cif.gz Display(77.67 KB)
5sjp_validation.cif
XML5sjp_validation.xml.gz Display(61.00 KB)
5sjp_validation.xml
PNG5sjp_multipercentile_validation.png.gz Display(167.46 KB)
5sjp_multipercentile_validation.png
SVG5sjp_multipercentile_validation.svg.gz Display(978.00 B)
5sjp_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5sjp_validation_2fo-fc_map_coef.cif.gz Display(1.10 MB)
5sjp_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5sjp_validation_fo-fc_map_coef.cif.gz Display(1.10 MB)
5sjp_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5sjp_validation_2fo-fc_map_coef.mtz Visualize(1.74 MB)
fo-fc (MTZ)5sjp_validation_fo-fc_map_coef.mtz Visualize(1.74 MB)

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PDB entries from 2026-01-14

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