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5SIY

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH c1(cc(nc2cc(nn12)c3c(nc4c(n3)cccc4)C)N5C[C@@H](CC5)F)N(C6CCOCC6)C, micromolar IC50=0.0050385

Resources
File formatFile name (file size)
PDBx/mmCIF5siy.cif.gz Display(274.79 KB)
5siy.cif
PDBx/mmJSONall5siy.json.gz Display (Tree)(170.15 KB)
5siy.json
no-atom5siy-noatom.json.gz Display (Header)(20.29 KB)
5siy-noatom.json
add only5siy-plus.json.gz Display(1.05 KB)
5siy-plus.json
PDBMLall5siy.xml.gz Display(376.85 KB)
5siy.xml
no-atom5siy-noatom.xml.gz Display(55.37 KB)
5siy-noatom.xml
ext-atom5siy-extatom.xml.gz Display(242.36 KB)
5siy-extatom.xml
pdb_nextgenallpdb_00005siy_xyz-enrich.cif.gz Display(300.14 KB)
pdb_00005siy_xyz-enrich.cif
no-atompdb_00005siy_xyz-no-atom-enrich.xml.gz Display(68.40 KB)
pdb_00005siy_xyz-no-atom-enrich.xml
ng-only5siy-plus.json.gz Display(3.41 KB)
5siy-plus.json
PDBpdb5siy.ent.gz Display(221.05 KB)
pdb5siy.ent
RDF5siy.rdf.gz Visualize(151.01 KB)
5siy.rdf
Structure factorsr5siysf.ent.gz Display(13.54 MB)
r5siysf.ent
Biological unit (mmCIF format)5siy-assembly1.cif.gz Display(70.80 KB)
5siy-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5siy-assembly2.cif.gz Display(71.74 KB)
5siy-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

5siy-assembly3.cif.gz Display(71.73 KB)
5siy-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

5siy-assembly4.cif.gz Display(69.36 KB)
5siy-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5siy.pdb1.gz Display(56.19 KB)
5siy.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5siy.pdb2.gz Display(56.54 KB)
5siy.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

5siy.pdb3.gz Display(57.01 KB)
5siy.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

5siy.pdb4.gz Display(55.22 KB)
5siy.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5siy_validation.pdf.gz Display(1.52 MB)
5siy_validation.pdf
PDF-full5siy_full_validation.pdf.gz Display(1.54 MB)
5siy_full_validation.pdf
mmCIF5siy_validation.cif.gz Display(77.23 KB)
5siy_validation.cif
XML5siy_validation.xml.gz Display(60.40 KB)
5siy_validation.xml
PNG5siy_multipercentile_validation.png.gz Display(165.23 KB)
5siy_multipercentile_validation.png
SVG5siy_multipercentile_validation.svg.gz Display(953.00 B)
5siy_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5siy_validation_2fo-fc_map_coef.cif.gz Display(1.51 MB)
5siy_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5siy_validation_fo-fc_map_coef.cif.gz Display(1.50 MB)
5siy_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5siy_validation_2fo-fc_map_coef.mtz Visualize(2.38 MB)
fo-fc (MTZ)5siy_validation_fo-fc_map_coef.mtz Visualize(2.38 MB)

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PDB entries from 2026-01-21

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