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5SIS

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH c1(c(n(nc1)C)C(Nc3cc2nc(cn2cc3)c4ccccc4)=O)C(=O)N(C)CCNC, micromolar IC50=0.002096

Resources
File formatFile name (file size)
PDBx/mmCIF5sis.cif.gz Display(88.75 KB)
5sis.cif
PDBx/mmJSONall5sis.json.gz Display (Tree)(63.52 KB)
5sis.json
no-atom5sis-noatom.json.gz Display (Header)(17.31 KB)
5sis-noatom.json
add only5sis-plus.json.gz Display(849.00 B)
5sis-plus.json
PDBMLall5sis.xml.gz Display(118.11 KB)
5sis.xml
no-atom5sis-noatom.xml.gz Display(30.68 KB)
5sis-noatom.xml
ext-atom5sis-extatom.xml.gz Display(66.23 KB)
5sis-extatom.xml
pdb_nextgenallpdb_00005sis_xyz-enrich.cif.gz Display(96.70 KB)
pdb_00005sis_xyz-enrich.cif
no-atompdb_00005sis_xyz-no-atom-enrich.xml.gz Display(34.49 KB)
pdb_00005sis_xyz-no-atom-enrich.xml
ng-only5sis-plus.json.gz Display(2.84 KB)
5sis-plus.json
PDBpdb5sis.ent.gz Display(65.16 KB)
pdb5sis.ent
RDF5sis.rdf.gz Visualize(85.48 KB)
5sis.rdf
Structure factorsr5sissf.ent.gz Display(5.23 MB)
r5sissf.ent
Biological unit (mmCIF format)5sis-assembly1.cif.gz Display(76.71 KB)
5sis-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5sis.pdb1.gz Display(59.51 KB)
5sis.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5sis_validation.pdf.gz Display(699.29 KB)
5sis_validation.pdf
PDF-full5sis_full_validation.pdf.gz Display(700.60 KB)
5sis_full_validation.pdf
mmCIF5sis_validation.cif.gz Display(26.84 KB)
5sis_validation.cif
XML5sis_validation.xml.gz Display(18.72 KB)
5sis_validation.xml
PNG5sis_multipercentile_validation.png.gz Display(158.49 KB)
5sis_multipercentile_validation.png
SVG5sis_multipercentile_validation.svg.gz Display(917.00 B)
5sis_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5sis_validation_2fo-fc_map_coef.cif.gz Display(583.44 KB)
5sis_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5sis_validation_fo-fc_map_coef.cif.gz Display(581.77 KB)
5sis_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5sis_validation_2fo-fc_map_coef.mtz Visualize(948.61 KB)
fo-fc (MTZ)5sis_validation_fo-fc_map_coef.mtz Visualize(948.61 KB)

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PDB entries from 2026-01-14

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