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5SIR

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH c1c(C)nc(c(c1)C)C(=O)Nc3nc2nc(cn2cc3)c4ccccc4, micromolar IC50=0.028279

Resources
File formatFile name (file size)
PDBx/mmCIF5sir.cif.gz Display(270.69 KB)
5sir.cif
PDBx/mmJSONall5sir.json.gz Display (Tree)(166.41 KB)
5sir.json
no-atom5sir-noatom.json.gz Display (Header)(19.83 KB)
5sir-noatom.json
add only5sir-plus.json.gz Display(1015.00 B)
5sir-plus.json
PDBMLall5sir.xml.gz Display(370.39 KB)
5sir.xml
no-atom5sir-noatom.xml.gz Display(54.22 KB)
5sir-noatom.xml
ext-atom5sir-extatom.xml.gz Display(239.33 KB)
5sir-extatom.xml
pdb_nextgenallpdb_00005sir_xyz-enrich.cif.gz Display(295.86 KB)
pdb_00005sir_xyz-enrich.cif
no-atompdb_00005sir_xyz-no-atom-enrich.xml.gz Display(67.35 KB)
pdb_00005sir_xyz-no-atom-enrich.xml
ng-only5sir-plus.json.gz Display(3.42 KB)
5sir-plus.json
PDBpdb5sir.ent.gz Display(217.97 KB)
pdb5sir.ent
RDF5sir.rdf.gz Visualize(148.15 KB)
5sir.rdf
Structure factorsr5sirsf.ent.gz Display(4.43 MB)
r5sirsf.ent
Biological unit (mmCIF format)5sir-assembly1.cif.gz Display(70.24 KB)
5sir-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5sir-assembly2.cif.gz Display(70.56 KB)
5sir-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

5sir-assembly3.cif.gz Display(69.26 KB)
5sir-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

5sir-assembly4.cif.gz Display(68.61 KB)
5sir-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5sir.pdb1.gz Display(56.07 KB)
5sir.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5sir.pdb2.gz Display(55.86 KB)
5sir.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

5sir.pdb3.gz Display(55.43 KB)
5sir.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

5sir.pdb4.gz Display(54.86 KB)
5sir.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5sir_validation.pdf.gz Display(1.20 MB)
5sir_validation.pdf
PDF-full5sir_full_validation.pdf.gz Display(1.22 MB)
5sir_full_validation.pdf
mmCIF5sir_validation.cif.gz Display(70.64 KB)
5sir_validation.cif
XML5sir_validation.xml.gz Display(53.45 KB)
5sir_validation.xml
PNG5sir_multipercentile_validation.png.gz Display(161.77 KB)
5sir_multipercentile_validation.png
SVG5sir_multipercentile_validation.svg.gz Display(956.00 B)
5sir_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5sir_validation_2fo-fc_map_coef.cif.gz Display(857.45 KB)
5sir_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5sir_validation_fo-fc_map_coef.cif.gz Display(862.62 KB)
5sir_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5sir_validation_2fo-fc_map_coef.mtz Visualize(1.30 MB)
fo-fc (MTZ)5sir_validation_fo-fc_map_coef.mtz Visualize(1.30 MB)

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PDB entries from 2026-01-14

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