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5SIP

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH c1(c(n(nc1)C)C(=O)Nc3nc2nc(cn2cc3)c4ccccc4)C(N5CCC5)=O, micromolar IC50=0.0027158

Resources
File formatFile name (file size)
PDBx/mmCIF5sip.cif.gz Display(274.66 KB)
5sip.cif
PDBx/mmJSONall5sip.json.gz Display (Tree)(169.97 KB)
5sip.json
no-atom5sip-noatom.json.gz Display (Header)(20.14 KB)
5sip-noatom.json
add only5sip-plus.json.gz Display(1014.00 B)
5sip-plus.json
PDBMLall5sip.xml.gz Display(375.74 KB)
5sip.xml
no-atom5sip-noatom.xml.gz Display(55.01 KB)
5sip-noatom.xml
ext-atom5sip-extatom.xml.gz Display(242.44 KB)
5sip-extatom.xml
pdb_nextgenallpdb_00005sip_xyz-enrich.cif.gz Display(299.95 KB)
pdb_00005sip_xyz-enrich.cif
no-atompdb_00005sip_xyz-no-atom-enrich.xml.gz Display(67.58 KB)
pdb_00005sip_xyz-no-atom-enrich.xml
ng-only5sip-plus.json.gz Display(3.42 KB)
5sip-plus.json
PDBpdb5sip.ent.gz Display(220.70 KB)
pdb5sip.ent
RDF5sip.rdf.gz Visualize(149.81 KB)
5sip.rdf
Structure factorsr5sipsf.ent.gz Display(13.26 MB)
r5sipsf.ent
Biological unit (mmCIF format)5sip-assembly1.cif.gz Display(71.11 KB)
5sip-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5sip-assembly2.cif.gz Display(71.90 KB)
5sip-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

5sip-assembly3.cif.gz Display(71.94 KB)
5sip-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

5sip-assembly4.cif.gz Display(69.03 KB)
5sip-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5sip.pdb1.gz Display(56.46 KB)
5sip.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5sip.pdb2.gz Display(56.76 KB)
5sip.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

5sip.pdb3.gz Display(57.14 KB)
5sip.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

5sip.pdb4.gz Display(54.80 KB)
5sip.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5sip_validation.pdf.gz Display(1.36 MB)
5sip_validation.pdf
PDF-full5sip_full_validation.pdf.gz Display(1.37 MB)
5sip_full_validation.pdf
mmCIF5sip_validation.cif.gz Display(74.99 KB)
5sip_validation.cif
XML5sip_validation.xml.gz Display(57.75 KB)
5sip_validation.xml
PNG5sip_multipercentile_validation.png.gz Display(168.06 KB)
5sip_multipercentile_validation.png
SVG5sip_multipercentile_validation.svg.gz Display(954.00 B)
5sip_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5sip_validation_2fo-fc_map_coef.cif.gz Display(1.51 MB)
5sip_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5sip_validation_fo-fc_map_coef.cif.gz Display(1.51 MB)
5sip_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5sip_validation_2fo-fc_map_coef.mtz Visualize(2.38 MB)
fo-fc (MTZ)5sip_validation_fo-fc_map_coef.mtz Visualize(2.38 MB)

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PDB entries from 2025-07-09

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