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5SIM

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH C(=O)(N1CCCC1C)c5c(C(Nc3cc2nc(cn2cc3)c4ccccc4)=O)n(nc5)C, micromolar IC50=0.000107

Resources
File formatFile name (file size)
PDBx/mmCIF5sim.cif.gz Display(88.81 KB)
5sim.cif
PDBx/mmJSONall5sim.json.gz Display (Tree)(63.95 KB)
5sim.json
no-atom5sim-noatom.json.gz Display (Header)(17.08 KB)
5sim-noatom.json
add only5sim-plus.json.gz Display(856.00 B)
5sim-plus.json
PDBMLall5sim.xml.gz Display(119.20 KB)
5sim.xml
no-atom5sim-noatom.xml.gz Display(30.42 KB)
5sim-noatom.xml
ext-atom5sim-extatom.xml.gz Display(66.93 KB)
5sim-extatom.xml
pdb_nextgenallpdb_00005sim_xyz-enrich.cif.gz Display(96.73 KB)
pdb_00005sim_xyz-enrich.cif
no-atompdb_00005sim_xyz-no-atom-enrich.xml.gz Display(33.91 KB)
pdb_00005sim_xyz-no-atom-enrich.xml
ng-only5sim-plus.json.gz Display(2.84 KB)
5sim-plus.json
PDBpdb5sim.ent.gz Display(65.67 KB)
pdb5sim.ent
RDF5sim.rdf.gz Visualize(85.08 KB)
5sim.rdf
Structure factorsr5simsf.ent.gz Display(6.75 MB)
r5simsf.ent
Biological unit (mmCIF format)5sim-assembly1.cif.gz Display(76.83 KB)
5sim-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5sim.pdb1.gz Display(59.91 KB)
5sim.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5sim_validation.pdf.gz Display(685.33 KB)
5sim_validation.pdf
PDF-full5sim_full_validation.pdf.gz Display(688.51 KB)
5sim_full_validation.pdf
mmCIF5sim_validation.cif.gz Display(26.65 KB)
5sim_validation.cif
XML5sim_validation.xml.gz Display(18.71 KB)
5sim_validation.xml
PNG5sim_multipercentile_validation.png.gz Display(162.08 KB)
5sim_multipercentile_validation.png
SVG5sim_multipercentile_validation.svg.gz Display(922.00 B)
5sim_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5sim_validation_2fo-fc_map_coef.cif.gz Display(685.55 KB)
5sim_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5sim_validation_fo-fc_map_coef.cif.gz Display(684.85 KB)
5sim_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5sim_validation_2fo-fc_map_coef.mtz Visualize(1.10 MB)
fo-fc (MTZ)5sim_validation_fo-fc_map_coef.mtz Visualize(1.10 MB)

238268

PDB entries from 2025-07-02

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