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5SIG

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH C1(NC(=Nc2c1cccc2)CN(C(=O)Nc3ccccc3)Cc4ccc(OC)cc4)=O, micromolar IC50=0.024784

Resources
File formatFile name (file size)
PDBx/mmCIF5sig.cif.gz Display(274.52 KB)
5sig.cif
PDBx/mmJSONall5sig.json.gz Display (Tree)(170.07 KB)
5sig.json
no-atom5sig-noatom.json.gz Display (Header)(20.13 KB)
5sig-noatom.json
add only5sig-plus.json.gz Display(1014.00 B)
5sig-plus.json
PDBMLall5sig.xml.gz Display(376.26 KB)
5sig.xml
no-atom5sig-noatom.xml.gz Display(55.16 KB)
5sig-noatom.xml
ext-atom5sig-extatom.xml.gz Display(243.08 KB)
5sig-extatom.xml
pdb_nextgenallpdb_00005sig_xyz-enrich.cif.gz Display(300.07 KB)
pdb_00005sig_xyz-enrich.cif
no-atompdb_00005sig_xyz-no-atom-enrich.xml.gz Display(68.18 KB)
pdb_00005sig_xyz-no-atom-enrich.xml
ng-only5sig-plus.json.gz Display(3.42 KB)
5sig-plus.json
PDBpdb5sig.ent.gz Display(221.23 KB)
pdb5sig.ent
RDF5sig.rdf.gz Visualize(150.07 KB)
5sig.rdf
Structure factorsr5sigsf.ent.gz Display(12.47 MB)
r5sigsf.ent
Biological unit (mmCIF format)5sig-assembly1.cif.gz Display(71.28 KB)
5sig-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5sig-assembly2.cif.gz Display(71.89 KB)
5sig-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

5sig-assembly3.cif.gz Display(71.33 KB)
5sig-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

5sig-assembly4.cif.gz Display(68.52 KB)
5sig-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5sig.pdb1.gz Display(56.95 KB)
5sig.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5sig.pdb2.gz Display(57.14 KB)
5sig.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

5sig.pdb3.gz Display(56.38 KB)
5sig.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

5sig.pdb4.gz Display(54.85 KB)
5sig.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5sig_validation.pdf.gz Display(1.42 MB)
5sig_validation.pdf
PDF-full5sig_full_validation.pdf.gz Display(1.43 MB)
5sig_full_validation.pdf
mmCIF5sig_validation.cif.gz Display(73.00 KB)
5sig_validation.cif
XML5sig_validation.xml.gz Display(55.19 KB)
5sig_validation.xml
PNG5sig_multipercentile_validation.png.gz Display(164.12 KB)
5sig_multipercentile_validation.png
SVG5sig_multipercentile_validation.svg.gz Display(923.00 B)
5sig_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5sig_validation_2fo-fc_map_coef.cif.gz Display(1.56 MB)
5sig_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5sig_validation_fo-fc_map_coef.cif.gz Display(1.55 MB)
5sig_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5sig_validation_2fo-fc_map_coef.mtz Visualize(2.37 MB)
fo-fc (MTZ)5sig_validation_fo-fc_map_coef.mtz Visualize(2.37 MB)

246704

PDB entries from 2025-12-24

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