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5SI8

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH c1(cn(nc1C(=O)Nc3cc2nc(cn2cc3C#N)c4ccccc4)C)C(=O)N5CCOCC5, micromolar IC50=0.060125

Resources
File formatFile name (file size)
PDBx/mmCIF5si8.cif.gz Display(273.19 KB)
5si8.cif
PDBx/mmJSONall5si8.json.gz Display (Tree)(168.36 KB)
5si8.json
no-atom5si8-noatom.json.gz Display (Header)(20.02 KB)
5si8-noatom.json
add only5si8-plus.json.gz Display(1014.00 B)
5si8-plus.json
PDBMLall5si8.xml.gz Display(373.72 KB)
5si8.xml
no-atom5si8-noatom.xml.gz Display(54.79 KB)
5si8-noatom.xml
ext-atom5si8-extatom.xml.gz Display(241.43 KB)
5si8-extatom.xml
pdb_nextgenallpdb_00005si8_xyz-enrich.cif.gz Display(298.50 KB)
pdb_00005si8_xyz-enrich.cif
no-atompdb_00005si8_xyz-no-atom-enrich.xml.gz Display(67.35 KB)
pdb_00005si8_xyz-no-atom-enrich.xml
ng-only5si8-plus.json.gz Display(3.42 KB)
5si8-plus.json
PDBpdb5si8.ent.gz Display(220.30 KB)
pdb5si8.ent
RDF5si8.rdf.gz Visualize(149.55 KB)
5si8.rdf
Structure factorsr5si8sf.ent.gz Display(4.18 MB)
r5si8sf.ent
Biological unit (mmCIF format)5si8-assembly1.cif.gz Display(71.17 KB)
5si8-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5si8-assembly2.cif.gz Display(71.25 KB)
5si8-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

5si8-assembly3.cif.gz Display(71.38 KB)
5si8-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

5si8-assembly4.cif.gz Display(68.88 KB)
5si8-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5si8.pdb1.gz Display(56.49 KB)
5si8.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5si8.pdb2.gz Display(56.54 KB)
5si8.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

5si8.pdb3.gz Display(56.74 KB)
5si8.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

5si8.pdb4.gz Display(54.91 KB)
5si8.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5si8_validation.pdf.gz Display(1.35 MB)
5si8_validation.pdf
PDF-full5si8_full_validation.pdf.gz Display(1.36 MB)
5si8_full_validation.pdf
mmCIF5si8_validation.cif.gz Display(74.66 KB)
5si8_validation.cif
XML5si8_validation.xml.gz Display(58.09 KB)
5si8_validation.xml
PNG5si8_multipercentile_validation.png.gz Display(169.42 KB)
5si8_multipercentile_validation.png
SVG5si8_multipercentile_validation.svg.gz Display(983.00 B)
5si8_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5si8_validation_2fo-fc_map_coef.cif.gz Display(1.16 MB)
5si8_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5si8_validation_fo-fc_map_coef.cif.gz Display(1.15 MB)
5si8_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5si8_validation_2fo-fc_map_coef.mtz Visualize(2.14 MB)
fo-fc (MTZ)5si8_validation_fo-fc_map_coef.mtz Visualize(2.14 MB)

238895

PDB entries from 2025-07-16

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