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5SI4

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH C1=CN(N=C(C1=O)c2ccnn2c3c4c(ccc3)cccc4)c5cc(ccc5)OC(F)(F)F, micromolar IC50=0.002773

Resources
File formatFile name (file size)
PDBx/mmCIF5si4.cif.gz Display(278.61 KB)
5si4.cif
PDBx/mmJSONall5si4.json.gz Display (Tree)(172.32 KB)
5si4.json
no-atom5si4-noatom.json.gz Display (Header)(20.59 KB)
5si4-noatom.json
add only5si4-plus.json.gz Display(1015.00 B)
5si4-plus.json
PDBMLall5si4.xml.gz Display(380.48 KB)
5si4.xml
no-atom5si4-noatom.xml.gz Display(55.49 KB)
5si4-noatom.xml
ext-atom5si4-extatom.xml.gz Display(246.11 KB)
5si4-extatom.xml
pdb_nextgenallpdb_00005si4_xyz-enrich.cif.gz Display(304.06 KB)
pdb_00005si4_xyz-enrich.cif
no-atompdb_00005si4_xyz-no-atom-enrich.xml.gz Display(68.67 KB)
pdb_00005si4_xyz-no-atom-enrich.xml
ng-only5si4-plus.json.gz Display(3.41 KB)
5si4-plus.json
PDBpdb5si4.ent.gz Display(225.85 KB)
pdb5si4.ent
RDF5si4.rdf.gz Visualize(150.61 KB)
5si4.rdf
Structure factorsr5si4sf.ent.gz Display(7.88 MB)
r5si4sf.ent
Biological unit (mmCIF format)5si4-assembly1.cif.gz Display(72.53 KB)
5si4-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5si4-assembly2.cif.gz Display(72.70 KB)
5si4-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

5si4-assembly3.cif.gz Display(72.99 KB)
5si4-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

5si4-assembly4.cif.gz Display(69.50 KB)
5si4-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5si4.pdb1.gz Display(57.78 KB)
5si4.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5si4.pdb2.gz Display(57.85 KB)
5si4.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

5si4.pdb3.gz Display(57.98 KB)
5si4.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

5si4.pdb4.gz Display(55.41 KB)
5si4.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5si4_validation.pdf.gz Display(2.49 MB)
5si4_validation.pdf
PDF-full5si4_full_validation.pdf.gz Display(2.51 MB)
5si4_full_validation.pdf
mmCIF5si4_validation.cif.gz Display(75.81 KB)
5si4_validation.cif
XML5si4_validation.xml.gz Display(58.15 KB)
5si4_validation.xml
PNG5si4_multipercentile_validation.png.gz Display(169.51 KB)
5si4_multipercentile_validation.png
SVG5si4_multipercentile_validation.svg.gz Display(956.00 B)
5si4_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5si4_validation_2fo-fc_map_coef.cif.gz Display(974.23 KB)
5si4_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5si4_validation_fo-fc_map_coef.cif.gz Display(970.58 KB)
5si4_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5si4_validation_2fo-fc_map_coef.mtz Visualize(1.47 MB)
fo-fc (MTZ)5si4_validation_fo-fc_map_coef.mtz Visualize(1.47 MB)

240971

PDB entries from 2025-08-27

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