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5SHZ

CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH C2(=NN(c1ccccc1)C=CC2=O)c3ccnn3c4cccc(c4)C#C, micromolar IC50=0.004957

Resources
File formatFile name (file size)
PDBx/mmCIF5shz.cif.gz Display(264.12 KB)
5shz.cif
PDBx/mmJSONall5shz.json.gz Display (Tree)(162.03 KB)
5shz.json
no-atom5shz-noatom.json.gz Display (Header)(17.89 KB)
5shz-noatom.json
add only5shz-plus.json.gz Display(1.08 KB)
5shz-plus.json
PDBMLall5shz.xml.gz Display(361.17 KB)
5shz.xml
no-atom5shz-noatom.xml.gz Display(49.63 KB)
5shz-noatom.xml
ext-atom5shz-extatom.xml.gz Display(236.02 KB)
5shz-extatom.xml
pdb_nextgenallpdb_00005shz_xyz-enrich.cif.gz Display(288.75 KB)
pdb_00005shz_xyz-enrich.cif
no-atompdb_00005shz_xyz-no-atom-enrich.xml.gz Display(65.13 KB)
pdb_00005shz_xyz-no-atom-enrich.xml
ng-only5shz-plus.json.gz Display(3.66 KB)
5shz-plus.json
PDBpdb5shz.ent.gz Display(215.01 KB)
pdb5shz.ent
RDF5shz.rdf.gz Visualize(140.61 KB)
5shz.rdf
Structure factorsr5shzsf.ent.gz Display(5.96 MB)
r5shzsf.ent
Biological unit (mmCIF format)5shz-assembly1.cif.gz Display(68.46 KB)
5shz-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

5shz-assembly2.cif.gz Display(69.33 KB)
5shz-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

5shz-assembly3.cif.gz Display(68.51 KB)
5shz-assembly3.cif (C)

*author defined assembly, 1 molecule(s) (monomeric)

5shz-assembly4.cif.gz Display(67.86 KB)
5shz-assembly4.cif (D)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5shz.pdb1.gz Display(54.71 KB)
5shz.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

5shz.pdb2.gz Display(55.36 KB)
5shz.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

5shz.pdb3.gz Display(54.80 KB)
5shz.pdb3 (C)

*author defined assembly, 1 molecule(s) (monomeric)

5shz.pdb4.gz Display(54.20 KB)
5shz.pdb4 (D)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5shz_validation.pdf.gz Display(1.74 MB)
5shz_validation.pdf
PDF-full5shz_full_validation.pdf.gz Display(1.75 MB)
5shz_full_validation.pdf
mmCIF5shz_validation.cif.gz Display(66.58 KB)
5shz_validation.cif
XML5shz_validation.xml.gz Display(51.71 KB)
5shz_validation.xml
PNG5shz_multipercentile_validation.png.gz Display(168.13 KB)
5shz_multipercentile_validation.png
SVG5shz_multipercentile_validation.svg.gz Display(981.00 B)
5shz_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5shz_validation_2fo-fc_map_coef.cif.gz Display(769.88 KB)
5shz_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5shz_validation_fo-fc_map_coef.cif.gz Display(765.79 KB)
5shz_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5shz_validation_2fo-fc_map_coef.mtz Visualize(1.20 MB)
fo-fc (MTZ)5shz_validation_fo-fc_map_coef.mtz Visualize(1.20 MB)

250359

PDB entries from 2026-03-11

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