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5MW3

Crystal structure of Dot1L in complex with inhibitor CPD1 [N6-(2,6-dichlorophenyl)-N6-(pent-2-yn-1-yl)quinoline-4,6-diamine] and inhibitor CPD2 [(R)-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-3-amine]

Resources
File formatFile name (file size)
PDBx/mmCIF5mw3.cif.gz Display(278.85 KB)
5mw3.cif
PDBx/mmJSONall5mw3.json.gz Display (Tree)(188.62 KB)
5mw3.json
no-atom5mw3-noatom.json.gz Display (Header)(17.17 KB)
5mw3-noatom.json
add only5mw3-plus.json.gz Display(985.00 B)
5mw3-plus.json
PDBMLall5mw3.xml.gz Display(384.92 KB)
5mw3.xml
no-atom5mw3-noatom.xml.gz Display(37.31 KB)
5mw3-noatom.xml
ext-atom5mw3-extatom.xml.gz Display(125.61 KB)
5mw3-extatom.xml
PDBpdb5mw3.ent.gz Display(225.58 KB)
pdb5mw3.ent
RDF5mw3.rdf.gz Visualize(108.02 KB)
5mw3.rdf
Structure factorsr5mw3sf.ent.gz Display(527.03 KB)
r5mw3sf.ent
Biological unit (mmCIF format)5mw3-assembly1.cif.gz Display(139.14 KB)
5mw3-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

5mw3-assembly2.cif.gz Display(138.50 KB)
5mw3-assembly2.cif (B)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5mw3.pdb1.gz Display(111.56 KB)
5mw3.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

5mw3.pdb2.gz Display(111.87 KB)
5mw3.pdb2 (B)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5mw3_validation.pdf.gz Display(1.18 MB)
5mw3_validation.pdf
PDF-full5mw3_full_validation.pdf.gz Display(1.19 MB)
5mw3_full_validation.pdf
mmCIF5mw3_validation.cif.gz Display(41.20 KB)
5mw3_validation.cif
XML5mw3_validation.xml.gz Display(28.42 KB)
5mw3_validation.xml
PNG5mw3_multipercentile_validation.png.gz Display(154.37 KB)
5mw3_multipercentile_validation.png
SVG5mw3_multipercentile_validation.svg.gz Display(920.00 B)
5mw3_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5mw3_validation_2fo-fc_map_coef.cif.gz Display(920.60 KB)
5mw3_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5mw3_validation_fo-fc_map_coef.cif.gz Display(919.77 KB)
5mw3_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5mw3_validation_2fo-fc_map_coef.mtz Visualize(1.44 MB)
fo-fc (MTZ)5mw3_validation_fo-fc_map_coef.mtz Visualize(1.44 MB)

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PDB entries from 2024-07-17

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