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5K7K

Design and Optimization of Biaryl Ether Aryl Sulfonamides as Selective Inhibitors of NaV1.7: Discovery of Clinical Candidate PF-05089771

Resources
File formatFile name (file size)
PDBx/mmCIF5k7k.cif.gz Display(110.85 KB)
5k7k.cif
PDBx/mmJSONall5k7k.json.gz Display (Tree)(78.33 KB)
5k7k.json
no-atom5k7k-noatom.json.gz Display (Header)(18.53 KB)
5k7k-noatom.json
add only5k7k-plus.json.gz Display(1.50 KB)
5k7k-plus.json
PDBMLall5k7k.xml.gz Display(145.18 KB)
5k7k.xml
no-atom5k7k-noatom.xml.gz Display(31.57 KB)
5k7k-noatom.xml
ext-atom5k7k-extatom.xml.gz Display(86.13 KB)
5k7k-extatom.xml
PDBpdb5k7k.ent.gz Display(83.15 KB)
pdb5k7k.ent
RDF5k7k.rdf.gz Visualize(95.89 KB)
5k7k.rdf
Structure factorsr5k7ksf.ent.gz Display(496.99 KB)
r5k7ksf.ent
Biological unit (mmCIF format)5k7k-assembly1.cif.gz Display(97.63 KB)
5k7k-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5k7k.pdb1.gz Display(77.07 KB)
5k7k.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5k7k_validation.pdf.gz Display(1.11 MB)
5k7k_validation.pdf
PDF-full5k7k_full_validation.pdf.gz Display(1.12 MB)
5k7k_full_validation.pdf
mmCIF5k7k_validation.cif.gz Display(26.74 KB)
5k7k_validation.cif
XML5k7k_validation.xml.gz Display(19.90 KB)
5k7k_validation.xml
PNG5k7k_multipercentile_validation.png.gz Display(168.47 KB)
5k7k_multipercentile_validation.png
SVG5k7k_multipercentile_validation.svg.gz Display(973.00 B)
5k7k_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5k7k_validation_2fo-fc_map_coef.cif.gz Display(246.36 KB)
5k7k_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5k7k_validation_fo-fc_map_coef.cif.gz Display(241.02 KB)
5k7k_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5k7k_validation_2fo-fc_map_coef.mtz Visualize(556.99 KB)
fo-fc (MTZ)5k7k_validation_fo-fc_map_coef.mtz Visualize(556.99 KB)

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PDB entries from 2024-07-24

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