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5IIS

Design, synthesis and structure activity relationship of potent pan-PIM kinase inhibitors derived from the pyridyl-amide scaffold

Resources
File formatFile name (file size)
PDBx/mmCIF5iis.cif.gz Display(103.19 KB)
5iis.cif
PDBx/mmJSONall5iis.json.gz Display (Tree)(69.08 KB)
5iis.json
no-atom5iis-noatom.json.gz Display (Header)(12.98 KB)
5iis-noatom.json
add only5iis-plus.json.gz Display(1.13 KB)
5iis-plus.json
PDBMLall5iis.xml.gz Display(148.29 KB)
5iis.xml
no-atom5iis-noatom.xml.gz Display(18.88 KB)
5iis-noatom.xml
ext-atom5iis-extatom.xml.gz Display(56.74 KB)
5iis-extatom.xml
PDBpdb5iis.ent.gz Display(79.19 KB)
pdb5iis.ent
RDF5iis.rdf.gz Visualize(44.26 KB)
5iis.rdf
Structure factorsr5iissf.ent.gz Display(713.63 KB)
r5iissf.ent
Biological unit (mmCIF format)5iis-assembly1.cif.gz Display(96.64 KB)
5iis-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5iis.pdb1.gz Display(74.69 KB)
5iis.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5iis_validation.pdf.gz Display(448.31 KB)
5iis_validation.pdf
PDF-full5iis_full_validation.pdf.gz Display(448.84 KB)
5iis_full_validation.pdf
mmCIF5iis_validation.cif.gz Display(20.62 KB)
5iis_validation.cif
XML5iis_validation.xml.gz Display(14.25 KB)
5iis_validation.xml
PNG5iis_multipercentile_validation.png.gz Display(159.59 KB)
5iis_multipercentile_validation.png
SVG5iis_multipercentile_validation.svg.gz Display(955.00 B)
5iis_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5iis_validation_2fo-fc_map_coef.cif.gz Display(370.24 KB)
5iis_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5iis_validation_fo-fc_map_coef.cif.gz Display(371.55 KB)
5iis_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5iis_validation_2fo-fc_map_coef.mtz Visualize(603.84 KB)
fo-fc (MTZ)5iis_validation_fo-fc_map_coef.mtz Visualize(603.84 KB)

224004

PDB entries from 2024-08-21

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