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5DWR

Identification of N-(4-((1R,3S,5S)-3-amino-5-methylcyclohexyl)pyridin-3-yl)-6-(2,6-difluorophenyl)-5-fluoropicolinamide (PIM447), a Potent and Selective Proviral Insertion Site of Moloney Murine Leukemia (PIM) 1,2 and 3 Kinase Inhibitor in Clinical Trials for Hematological Malignancies

Resources
File formatFile name (file size)
PDBx/mmCIF5dwr.cif.gz Display(75.06 KB)
5dwr.cif
PDBx/mmJSONall5dwr.json.gz Display (Tree)(54.30 KB)
5dwr.json
no-atom5dwr-noatom.json.gz Display (Header)(13.72 KB)
5dwr-noatom.json
add only5dwr-plus.json.gz Display(1.62 KB)
5dwr-plus.json
PDBMLall5dwr.xml.gz Display(96.96 KB)
5dwr.xml
no-atom5dwr-noatom.xml.gz Display(21.22 KB)
5dwr-noatom.xml
ext-atom5dwr-extatom.xml.gz Display(56.95 KB)
5dwr-extatom.xml
PDBpdb5dwr.ent.gz Display(57.54 KB)
pdb5dwr.ent
RDF5dwr.rdf.gz Visualize(51.97 KB)
5dwr.rdf
Structure factorsr5dwrsf.ent.gz Display(748.96 KB)
r5dwrsf.ent
Biological unit (mmCIF format)5dwr-assembly1.cif.gz Display(67.83 KB)
5dwr-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5dwr.pdb1.gz Display(52.98 KB)
5dwr.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5dwr_validation.pdf.gz Display(616.94 KB)
5dwr_validation.pdf
PDF-full5dwr_full_validation.pdf.gz Display(618.25 KB)
5dwr_full_validation.pdf
XML5dwr_validation.xml.gz Display(15.21 KB)
5dwr_validation.xml
PNG5dwr_multipercentile_validation.png.gz Display(138.44 KB)
5dwr_multipercentile_validation.png
SVG5dwr_multipercentile_validation.svg.gz Display(934.00 B)
5dwr_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5dwr_validation_2fo-fc_map_coef.cif.gz Display(297.99 KB)
5dwr_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5dwr_validation_fo-fc_map_coef.cif.gz Display(292.20 KB)
5dwr_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5dwr_validation_2fo-fc_map_coef.mtz Visualize(708.80 KB)
fo-fc (MTZ)5dwr_validation_fo-fc_map_coef.mtz Visualize(708.80 KB)

219140

PDB entries from 2024-05-01

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