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5DWR

Identification of N-(4-((1R,3S,5S)-3-amino-5-methylcyclohexyl)pyridin-3-yl)-6-(2,6-difluorophenyl)-5-fluoropicolinamide (PIM447), a Potent and Selective Proviral Insertion Site of Moloney Murine Leukemia (PIM) 1,2 and 3 Kinase Inhibitor in Clinical Trials for Hematological Malignancies

Resources
File formatFile name (file size)
PDBx/mmCIF5dwr.cif.gz Display(79.92 KB)
5dwr.cif
PDBx/mmJSONall5dwr.json.gz Display (Tree)(56.25 KB)
5dwr.json
no-atom5dwr-noatom.json.gz Display (Header)(16.46 KB)
5dwr-noatom.json
add only5dwr-plus.json.gz Display(1.67 KB)
5dwr-plus.json
PDBMLall5dwr.xml.gz Display(104.11 KB)
5dwr.xml
no-atom5dwr-noatom.xml.gz Display(28.39 KB)
5dwr-noatom.xml
ext-atom5dwr-extatom.xml.gz Display(56.95 KB)
5dwr-extatom.xml
pdb_nextgenallpdb_00005dwr_xyz-enrich.cif.gz Display(89.29 KB)
pdb_00005dwr_xyz-enrich.cif
no-atompdb_00005dwr_xyz-no-atom-enrich.xml.gz Display(39.41 KB)
pdb_00005dwr_xyz-no-atom-enrich.xml
ng-only5dwr-plus.json.gz Display(2.67 KB)
5dwr-plus.json
PDBpdb5dwr.ent.gz Display(56.77 KB)
pdb5dwr.ent
RDF5dwr.rdf.gz Visualize(83.27 KB)
5dwr.rdf
Structure factorsr5dwrsf.ent.gz Display(748.96 KB)
r5dwrsf.ent
Biological unit (mmCIF format)5dwr-assembly1.cif.gz Display(67.84 KB)
5dwr-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5dwr.pdb1.gz Display(51.77 KB)
5dwr.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5dwr_validation.pdf.gz Display(813.66 KB)
5dwr_validation.pdf
PDF-full5dwr_full_validation.pdf.gz Display(815.07 KB)
5dwr_full_validation.pdf
mmCIF5dwr_validation.cif.gz Display(21.73 KB)
5dwr_validation.cif
XML5dwr_validation.xml.gz Display(14.90 KB)
5dwr_validation.xml
PNG5dwr_multipercentile_validation.png.gz Display(164.03 KB)
5dwr_multipercentile_validation.png
SVG5dwr_multipercentile_validation.svg.gz Display(953.00 B)
5dwr_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5dwr_validation_2fo-fc_map_coef.cif.gz Display(440.74 KB)
5dwr_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5dwr_validation_fo-fc_map_coef.cif.gz Display(442.26 KB)
5dwr_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5dwr_validation_2fo-fc_map_coef.mtz Visualize(708.80 KB)
fo-fc (MTZ)5dwr_validation_fo-fc_map_coef.mtz Visualize(708.80 KB)

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PDB entries from 2026-01-14

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