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5A2S

Potent, selective and CNS-penetrant tetrasubstituted cyclopropane class IIa histone deacetylase (HDAC) inhibitors

Resources
File formatFile name (file size)
PDBx/mmCIF5a2s.cif.gz Display(153.44 KB)
5a2s.cif
PDBx/mmJSONall5a2s.json.gz Display (Tree)(100.71 KB)
5a2s.json
no-atom5a2s-noatom.json.gz Display (Header)(15.66 KB)
5a2s-noatom.json
add only5a2s-plus.json.gz Display(944.00 B)
5a2s-plus.json
PDBMLall5a2s.xml.gz Display(208.01 KB)
5a2s.xml
no-atom5a2s-noatom.xml.gz Display(37.26 KB)
5a2s-noatom.xml
ext-atom5a2s-extatom.xml.gz Display(129.48 KB)
5a2s-extatom.xml
pdb_nextgenallpdb_00005a2s_xyz-enrich.cif.gz Display(175.52 KB)
pdb_00005a2s_xyz-enrich.cif
no-atompdb_00005a2s_xyz-no-atom-enrich.xml.gz Display(63.04 KB)
pdb_00005a2s_xyz-no-atom-enrich.xml
ng-only5a2s-plus.json.gz Display(4.19 KB)
5a2s-plus.json
PDBpdb5a2s.ent.gz Display(119.84 KB)
pdb5a2s.ent
RDF5a2s.rdf.gz Visualize(108.75 KB)
5a2s.rdf
Structure factorsr5a2ssf.ent.gz Display(398.12 KB)
r5a2ssf.ent
Biological unit (mmCIF format)5a2s-assembly1.cif.gz Display(75.80 KB)
5a2s-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

5a2s-assembly2.cif.gz Display(75.91 KB)
5a2s-assembly2.cif (B)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)5a2s.pdb1.gz Display(58.68 KB)
5a2s.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

5a2s.pdb2.gz Display(59.27 KB)
5a2s.pdb2 (B)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF5a2s_validation.pdf.gz Display(850.64 KB)
5a2s_validation.pdf
PDF-full5a2s_full_validation.pdf.gz Display(856.67 KB)
5a2s_full_validation.pdf
mmCIF5a2s_validation.cif.gz Display(39.34 KB)
5a2s_validation.cif
XML5a2s_validation.xml.gz Display(28.44 KB)
5a2s_validation.xml
PNG5a2s_multipercentile_validation.png.gz Display(167.22 KB)
5a2s_multipercentile_validation.png
SVG5a2s_multipercentile_validation.svg.gz Display(974.00 B)
5a2s_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)5a2s_validation_2fo-fc_map_coef.cif.gz Display(207.31 KB)
5a2s_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)5a2s_validation_fo-fc_map_coef.cif.gz Display(201.91 KB)
5a2s_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)5a2s_validation_2fo-fc_map_coef.mtz Visualize(496.91 KB)
fo-fc (MTZ)5a2s_validation_fo-fc_map_coef.mtz Visualize(496.91 KB)

225158

PDB entries from 2024-09-18

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