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4X2I

Discovery of benzotriazolo diazepines as orally-active inhibitors of BET bromodomains: Crystal structure of BRD4 with CPI-13

Resources
File formatFile name (file size)
PDBx/mmCIF4x2i.cif.gz Display(77.05 KB)
4x2i.cif
PDBx/mmJSONall4x2i.json.gz Display (Tree)(55.42 KB)
4x2i.json
no-atom4x2i-noatom.json.gz Display (Header)(12.01 KB)
4x2i-noatom.json
add only4x2i-plus.json.gz Display(923.00 B)
4x2i-plus.json
PDBMLall4x2i.xml.gz Display(102.19 KB)
4x2i.xml
no-atom4x2i-noatom.xml.gz Display(19.92 KB)
4x2i-noatom.xml
ext-atom4x2i-extatom.xml.gz Display(28.63 KB)
4x2i-extatom.xml
PDBpdb4x2i.ent.gz Display(56.89 KB)
pdb4x2i.ent
RDF4x2i.rdf.gz Visualize(57.87 KB)
4x2i.rdf
Structure factorsr4x2isf.ent.gz Display(692.71 KB)
r4x2isf.ent
Biological unit (mmCIF format)4x2i-assembly1.cif.gz Display(67.11 KB)
4x2i-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)4x2i.pdb1.gz Display(51.75 KB)
4x2i.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF4x2i_validation.pdf.gz Display(567.93 KB)
4x2i_validation.pdf
PDF-full4x2i_full_validation.pdf.gz Display(569.02 KB)
4x2i_full_validation.pdf
XML4x2i_validation.xml.gz Display(9.96 KB)
4x2i_validation.xml
PNG4x2i_multipercentile_validation.png.gz Display(144.22 KB)
4x2i_multipercentile_validation.png
SVG4x2i_multipercentile_validation.svg.gz Display(928.00 B)
4x2i_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)4x2i_validation_2fo-fc_map_coef.cif.gz Display(392.45 KB)
4x2i_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)4x2i_validation_fo-fc_map_coef.cif.gz Display(372.16 KB)
4x2i_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)4x2i_validation_2fo-fc_map_coef.mtz Visualize(971.61 KB)
fo-fc (MTZ)4x2i_validation_fo-fc_map_coef.mtz Visualize(971.61 KB)

220472

PDB entries from 2024-05-29

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