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4V26

VER-246608, a novel pan-isoform ATP competitive inhibitor of pyruvate dehydrogenase kinase, disrupts Warburg metabolism and induces context- dependent cytostasis in cancer cells

Resources
File formatFile name (file size)
PDBx/mmCIF4v26.cif.gz Display(88.18 KB)
4v26.cif
PDBx/mmJSONall4v26.json.gz Display (Tree)(61.48 KB)
4v26.json
no-atom4v26-noatom.json.gz Display (Header)(14.82 KB)
4v26-noatom.json
add only4v26-plus.json.gz Display(1.27 KB)
4v26-plus.json
PDBMLall4v26.xml.gz Display(118.25 KB)
4v26.xml
no-atom4v26-noatom.xml.gz Display(29.49 KB)
4v26-noatom.xml
ext-atom4v26-extatom.xml.gz Display(66.84 KB)
4v26-extatom.xml
pdb_nextgenallpdb_00004v26_xyz-enrich.cif.gz Display(97.77 KB)
pdb_00004v26_xyz-enrich.cif
no-atompdb_00004v26_xyz-no-atom-enrich.xml.gz Display(39.13 KB)
pdb_00004v26_xyz-no-atom-enrich.xml
ng-only4v26-plus.json.gz Display(2.93 KB)
4v26-plus.json
PDBpdb4v26.ent.gz Display(65.98 KB)
pdb4v26.ent
RDF4v26.rdf.gz Visualize(90.23 KB)
4v26.rdf
Structure factorsr4v26sf.ent.gz Display(376.54 KB)
r4v26sf.ent
Biological unit (mmCIF format)4v26-assembly1.cif.gz Display(147.51 KB)
4v26-assembly1.cif (A)

*author and software defined assembly, 2 molecule(s) (dimeric)

Biological unit (PDB format)4v26.pdb1.gz Display(117.54 KB)
4v26.pdb1 (A)

*author and software defined assembly, 2 molecule(s) (dimeric)

Validation reportsPDF4v26_validation.pdf.gz Display(992.81 KB)
4v26_validation.pdf
PDF-full4v26_full_validation.pdf.gz Display(1002.35 KB)
4v26_full_validation.pdf
mmCIF4v26_validation.cif.gz Display(23.41 KB)
4v26_validation.cif
XML4v26_validation.xml.gz Display(16.60 KB)
4v26_validation.xml
PNG4v26_multipercentile_validation.png.gz Display(166.71 KB)
4v26_multipercentile_validation.png
SVG4v26_multipercentile_validation.svg.gz Display(974.00 B)
4v26_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)4v26_validation_2fo-fc_map_coef.cif.gz Display(290.09 KB)
4v26_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)4v26_validation_fo-fc_map_coef.cif.gz Display(289.79 KB)
4v26_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)4v26_validation_2fo-fc_map_coef.mtz Visualize(470.20 KB)
fo-fc (MTZ)4v26_validation_fo-fc_map_coef.mtz Visualize(470.20 KB)

225681

PDB entries from 2024-10-02

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