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4UWH

Discovery of (2S)-8-((3R)-3-Methylmorpholin-4-yl)-1-(3-methyl-2-oxo- butyl)-2-(trifluoromethyl)-3,4-dihydro-2H-pyrimido(1,2-a)pyrimidin-6- one: a Novel Potent and Selective Inhibitor of Vps34 for the Treatment of Solid Tumors

Resources
File formatFile name (file size)
PDBx/mmCIF4uwh.cif.gz Display(136.10 KB)
4uwh.cif
PDBx/mmJSONall4uwh.json.gz Display (Tree)(93.36 KB)
4uwh.json
no-atom4uwh-noatom.json.gz Display (Header)(18.50 KB)
4uwh-noatom.json
add only4uwh-plus.json.gz Display(974.00 B)
4uwh-plus.json
PDBMLall4uwh.xml.gz Display(182.92 KB)
4uwh.xml
no-atom4uwh-noatom.xml.gz Display(37.25 KB)
4uwh-noatom.xml
ext-atom4uwh-extatom.xml.gz Display(110.04 KB)
4uwh-extatom.xml
PDBpdb4uwh.ent.gz Display(103.13 KB)
pdb4uwh.ent
RDF4uwh.rdf.gz Visualize(108.49 KB)
4uwh.rdf
Structure factorsr4uwhsf.ent.gz Display(650.29 KB)
r4uwhsf.ent
Biological unit (mmCIF format)4uwh-assembly1.cif.gz Display(126.25 KB)
4uwh-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)4uwh.pdb1.gz Display(98.08 KB)
4uwh.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF4uwh_validation.pdf.gz Display(848.17 KB)
4uwh_validation.pdf
PDF-full4uwh_full_validation.pdf.gz Display(849.38 KB)
4uwh_full_validation.pdf
mmCIF4uwh_validation.cif.gz Display(36.31 KB)
4uwh_validation.cif
XML4uwh_validation.xml.gz Display(24.07 KB)
4uwh_validation.xml
PNG4uwh_multipercentile_validation.png.gz Display(162.88 KB)
4uwh_multipercentile_validation.png
SVG4uwh_multipercentile_validation.svg.gz Display(952.00 B)
4uwh_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)4uwh_validation_2fo-fc_map_coef.cif.gz Display(596.61 KB)
4uwh_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)4uwh_validation_fo-fc_map_coef.cif.gz Display(578.57 KB)
4uwh_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)4uwh_validation_2fo-fc_map_coef.mtz Visualize(1.40 MB)
fo-fc (MTZ)4uwh_validation_fo-fc_map_coef.mtz Visualize(1.40 MB)

222926

PDB entries from 2024-07-24

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