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4HY1

Pyrrolopyrimidine inhibitors of dna gyrase b and topoisomerase iv, part i: structure guided discovery and optimization of dual targeting agents with potent, broad-spectrum enzymatic activity.

Resources
File formatFile name (file size)
PDBx/mmCIF4hy1.cif.gz Display(146.68 KB)
4hy1.cif
PDBx/mmJSONall4hy1.json.gz Display (Tree)(97.17 KB)
4hy1.json
no-atom4hy1-noatom.json.gz Display (Header)(18.87 KB)
4hy1-noatom.json
add only4hy1-plus.json.gz Display(933.00 B)
4hy1-plus.json
PDBMLall4hy1.xml.gz Display(199.45 KB)
4hy1.xml
no-atom4hy1-noatom.xml.gz Display(40.56 KB)
4hy1-noatom.xml
ext-atom4hy1-extatom.xml.gz Display(118.67 KB)
4hy1-extatom.xml
PDBpdb4hy1.ent.gz Display(112.15 KB)
pdb4hy1.ent
RDF4hy1.rdf.gz Visualize(115.88 KB)
4hy1.rdf
Structure factorsr4hy1sf.ent.gz Display(900.04 KB)
r4hy1sf.ent
Biological unit (mmCIF format)4hy1-assembly1.cif.gz Display(86.99 KB)
4hy1-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

4hy1-assembly2.cif.gz Display(56.82 KB)
4hy1-assembly2.cif (B)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)4hy1.pdb1.gz Display(66.83 KB)
4hy1.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

4hy1.pdb2.gz Display(42.80 KB)
4hy1.pdb2 (B)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF4hy1_validation.pdf.gz Display(1.02 MB)
4hy1_validation.pdf
PDF-full4hy1_full_validation.pdf.gz Display(1.04 MB)
4hy1_full_validation.pdf
mmCIF4hy1_validation.cif.gz Display(46.27 KB)
4hy1_validation.cif
XML4hy1_validation.xml.gz Display(31.47 KB)
4hy1_validation.xml
PNG4hy1_multipercentile_validation.png.gz Display(168.59 KB)
4hy1_multipercentile_validation.png
SVG4hy1_multipercentile_validation.svg.gz Display(977.00 B)
4hy1_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)4hy1_validation_2fo-fc_map_coef.cif.gz Display(713.04 KB)
4hy1_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)4hy1_validation_fo-fc_map_coef.cif.gz Display(699.84 KB)
4hy1_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)4hy1_validation_2fo-fc_map_coef.mtz Visualize(1.63 MB)
fo-fc (MTZ)4hy1_validation_fo-fc_map_coef.mtz Visualize(1.63 MB)

222036

PDB entries from 2024-07-03

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