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4C66

Discovery of Epigenetic Regulator I-BET762: Lead Optimization to Afford a Clinical Candidate Inhibitor of the BET Bromodomains

Resources
File formatFile name (file size)
PDBx/mmCIF4c66.cif.gz Display(64.38 KB)
4c66.cif
PDBx/mmJSONall4c66.json.gz Display (Tree)(47.32 KB)
4c66.json
no-atom4c66-noatom.json.gz Display (Header)(7.74 KB)
4c66-noatom.json
add only4c66-plus.json.gz Display(927.00 B)
4c66-plus.json
PDBMLall4c66.xml.gz Display(85.68 KB)
4c66.xml
no-atom4c66-noatom.xml.gz Display(12.79 KB)
4c66-noatom.xml
ext-atom4c66-extatom.xml.gz Display(27.23 KB)
4c66-extatom.xml
PDBpdb4c66.ent.gz Display(51.72 KB)
pdb4c66.ent
RDF4c66.rdf.gz Visualize(27.66 KB)
4c66.rdf
Structure factorsr4c66sf.ent.gz Display(196.23 KB)
r4c66sf.ent
Biological unit (mmCIF format)4c66-assembly1.cif.gz Display(59.74 KB)
4c66-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)4c66.pdb1.gz Display(47.75 KB)
4c66.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF4c66_validation.pdf.gz Display(610.31 KB)
4c66_validation.pdf
PDF-full4c66_full_validation.pdf.gz Display(610.22 KB)
4c66_full_validation.pdf
XML4c66_validation.xml.gz Display(9.06 KB)
4c66_validation.xml
PNG4c66_multipercentile_validation.png.gz Display(148.27 KB)
4c66_multipercentile_validation.png
SVG4c66_multipercentile_validation.svg.gz Display(935.00 B)
4c66_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)4c66_validation_2fo-fc_map_coef.cif.gz Display(105.09 KB)
4c66_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)4c66_validation_fo-fc_map_coef.cif.gz Display(102.16 KB)
4c66_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)4c66_validation_2fo-fc_map_coef.mtz Visualize(256.77 KB)
fo-fc (MTZ)4c66_validation_fo-fc_map_coef.mtz Visualize(256.77 KB)

218853

PDB entries from 2024-04-24

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