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4C4J

Structure-based design of orally bioavailable pyrrolopyridine inhibitors of the mitotic kinase MPS1

Resources
File formatFile name (file size)
PDBx/mmCIF4c4j.cif.gz Display(121.00 KB)
4c4j.cif
PDBx/mmJSONall4c4j.json.gz Display (Tree)(86.03 KB)
4c4j.json
no-atom4c4j-noatom.json.gz Display (Header)(13.48 KB)
4c4j-noatom.json
add only4c4j-plus.json.gz Display(1.01 KB)
4c4j-plus.json
PDBMLall4c4j.xml.gz Display(162.57 KB)
4c4j.xml
no-atom4c4j-noatom.xml.gz Display(27.87 KB)
4c4j-noatom.xml
ext-atom4c4j-extatom.xml.gz Display(46.99 KB)
4c4j-extatom.xml
PDBpdb4c4j.ent.gz Display(92.09 KB)
pdb4c4j.ent
RDF4c4j.rdf.gz Visualize(83.21 KB)
4c4j.rdf
Structure factorsr4c4jsf.ent.gz Display(792.12 KB)
r4c4jsf.ent
Biological unit (mmCIF format)4c4j-assembly1.cif.gz Display(108.91 KB)
4c4j-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)4c4j.pdb1.gz Display(86.56 KB)
4c4j.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF4c4j_validation.pdf.gz Display(741.21 KB)
4c4j_validation.pdf
PDF-full4c4j_full_validation.pdf.gz Display(744.78 KB)
4c4j_full_validation.pdf
mmCIF4c4j_validation.cif.gz Display(15.33 KB)
4c4j_validation.cif
XML4c4j_validation.xml.gz Display(11.97 KB)
4c4j_validation.xml
PNG4c4j_multipercentile_validation.png.gz Display(171.07 KB)
4c4j_multipercentile_validation.png
SVG4c4j_multipercentile_validation.svg.gz Display(962.00 B)
4c4j_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)4c4j_validation_2fo-fc_map_coef.cif.gz Display(150.63 KB)
4c4j_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)4c4j_validation_fo-fc_map_coef.cif.gz Display(146.89 KB)
4c4j_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)4c4j_validation_2fo-fc_map_coef.mtz Visualize(359.10 KB)
fo-fc (MTZ)4c4j_validation_fo-fc_map_coef.mtz Visualize(359.10 KB)

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PDB entries from 2024-07-17

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