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4C4I

Structure-based design of orally bioavailable pyrrolopyridine inhibitors of the mitotic kinase MPS1

Resources
File formatFile name (file size)
PDBx/mmCIF4c4i.cif.gz Display(118.37 KB)
4c4i.cif
PDBx/mmJSONall4c4i.json.gz Display (Tree)(84.37 KB)
4c4i.json
no-atom4c4i-noatom.json.gz Display (Header)(13.54 KB)
4c4i-noatom.json
add only4c4i-plus.json.gz Display(1.00 KB)
4c4i-plus.json
PDBMLall4c4i.xml.gz Display(159.07 KB)
4c4i.xml
no-atom4c4i-noatom.xml.gz Display(27.84 KB)
4c4i-noatom.xml
ext-atom4c4i-extatom.xml.gz Display(46.04 KB)
4c4i-extatom.xml
PDBpdb4c4i.ent.gz Display(89.88 KB)
pdb4c4i.ent
RDF4c4i.rdf.gz Visualize(83.48 KB)
4c4i.rdf
Structure factorsr4c4isf.ent.gz Display(652.08 KB)
r4c4isf.ent
Biological unit (mmCIF format)4c4i-assembly1.cif.gz Display(106.10 KB)
4c4i-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)4c4i.pdb1.gz Display(84.06 KB)
4c4i.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF4c4i_validation.pdf.gz Display(736.15 KB)
4c4i_validation.pdf
PDF-full4c4i_full_validation.pdf.gz Display(738.76 KB)
4c4i_full_validation.pdf
mmCIF4c4i_validation.cif.gz Display(14.54 KB)
4c4i_validation.cif
XML4c4i_validation.xml.gz Display(11.41 KB)
4c4i_validation.xml
PNG4c4i_multipercentile_validation.png.gz Display(167.19 KB)
4c4i_multipercentile_validation.png
SVG4c4i_multipercentile_validation.svg.gz Display(954.00 B)
4c4i_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)4c4i_validation_2fo-fc_map_coef.cif.gz Display(182.09 KB)
4c4i_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)4c4i_validation_fo-fc_map_coef.cif.gz Display(181.53 KB)
4c4i_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)4c4i_validation_2fo-fc_map_coef.mtz Visualize(292.84 KB)
fo-fc (MTZ)4c4i_validation_fo-fc_map_coef.mtz Visualize(292.84 KB)

223532

PDB entries from 2024-08-07

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