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4C4H

Structure-based design of orally bioavailable pyrrolopyridine inhibitors of the mitotic kinase MPS1

Resources
File formatFile name (file size)
PDBx/mmCIF4c4h.cif.gz Display(117.02 KB)
4c4h.cif
PDBx/mmJSONall4c4h.json.gz Display (Tree)(83.42 KB)
4c4h.json
no-atom4c4h-noatom.json.gz Display (Header)(13.28 KB)
4c4h-noatom.json
add only4c4h-plus.json.gz Display(1.01 KB)
4c4h-plus.json
PDBMLall4c4h.xml.gz Display(156.77 KB)
4c4h.xml
no-atom4c4h-noatom.xml.gz Display(27.22 KB)
4c4h-noatom.xml
ext-atom4c4h-extatom.xml.gz Display(45.89 KB)
4c4h-extatom.xml
PDBpdb4c4h.ent.gz Display(88.71 KB)
pdb4c4h.ent
RDF4c4h.rdf.gz Visualize(82.56 KB)
4c4h.rdf
Structure factorsr4c4hsf.ent.gz Display(473.86 KB)
r4c4hsf.ent
Biological unit (mmCIF format)4c4h-assembly1.cif.gz Display(105.11 KB)
4c4h-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)4c4h.pdb1.gz Display(83.25 KB)
4c4h.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF4c4h_validation.pdf.gz Display(743.93 KB)
4c4h_validation.pdf
PDF-full4c4h_full_validation.pdf.gz Display(745.68 KB)
4c4h_full_validation.pdf
XML4c4h_validation.xml.gz Display(11.66 KB)
4c4h_validation.xml
PNG4c4h_multipercentile_validation.png.gz Display(146.13 KB)
4c4h_multipercentile_validation.png
SVG4c4h_multipercentile_validation.svg.gz Display(938.00 B)
4c4h_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)4c4h_validation_2fo-fc_map_coef.cif.gz Display(103.46 KB)
4c4h_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)4c4h_validation_fo-fc_map_coef.cif.gz Display(95.68 KB)
4c4h_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)4c4h_validation_2fo-fc_map_coef.mtz Visualize(246.81 KB)
fo-fc (MTZ)4c4h_validation_fo-fc_map_coef.mtz Visualize(246.81 KB)

218500

PDB entries from 2024-04-17

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