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4C4E

Structure-based design of orally bioavailable pyrrolopyridine inhibitors of the mitotic kinase MPS1

Resources
File formatFile name (file size)
PDBx/mmCIF4c4e.cif.gz Display(124.64 KB)
4c4e.cif
PDBx/mmJSONall4c4e.json.gz Display (Tree)(88.21 KB)
4c4e.json
no-atom4c4e-noatom.json.gz Display (Header)(14.56 KB)
4c4e-noatom.json
add only4c4e-plus.json.gz Display(1.02 KB)
4c4e-plus.json
PDBMLall4c4e.xml.gz Display(167.42 KB)
4c4e.xml
no-atom4c4e-noatom.xml.gz Display(29.57 KB)
4c4e-noatom.xml
ext-atom4c4e-extatom.xml.gz Display(49.71 KB)
4c4e-extatom.xml
PDBpdb4c4e.ent.gz Display(94.63 KB)
pdb4c4e.ent
RDF4c4e.rdf.gz Visualize(88.53 KB)
4c4e.rdf
Structure factorsr4c4esf.ent.gz Display(794.28 KB)
r4c4esf.ent
Biological unit (mmCIF format)4c4e-assembly1.cif.gz Display(111.33 KB)
4c4e-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)4c4e.pdb1.gz Display(88.55 KB)
4c4e.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF4c4e_validation.pdf.gz Display(1.15 MB)
4c4e_validation.pdf
PDF-full4c4e_full_validation.pdf.gz Display(1.16 MB)
4c4e_full_validation.pdf
mmCIF4c4e_validation.cif.gz Display(16.33 KB)
4c4e_validation.cif
XML4c4e_validation.xml.gz Display(12.50 KB)
4c4e_validation.xml
PNG4c4e_multipercentile_validation.png.gz Display(167.31 KB)
4c4e_multipercentile_validation.png
SVG4c4e_multipercentile_validation.svg.gz Display(975.00 B)
4c4e_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)4c4e_validation_2fo-fc_map_coef.cif.gz Display(140.65 KB)
4c4e_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)4c4e_validation_fo-fc_map_coef.cif.gz Display(137.34 KB)
4c4e_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)4c4e_validation_2fo-fc_map_coef.mtz Visualize(337.40 KB)
fo-fc (MTZ)4c4e_validation_fo-fc_map_coef.mtz Visualize(337.40 KB)

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PDB entries from 2024-07-17

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