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4AN9

Crystal structures of human MEK1 with carboxamide-based allosteric inhibitor XL518 (GDC-0973), or related analogs.

Resources
File formatFile name (file size)
PDBx/mmCIF4an9.cif.gz Display(71.91 KB)
4an9.cif
PDBx/mmJSONall4an9.json.gz Display (Tree)(49.95 KB)
4an9.json
no-atom4an9-noatom.json.gz Display (Header)(14.08 KB)
4an9-noatom.json
add only4an9-plus.json.gz Display(1.26 KB)
4an9-plus.json
PDBMLall4an9.xml.gz Display(95.03 KB)
4an9.xml
no-atom4an9-noatom.xml.gz Display(26.94 KB)
4an9-noatom.xml
ext-atom4an9-extatom.xml.gz Display(51.10 KB)
4an9-extatom.xml
PDBpdb4an9.ent.gz Display(52.17 KB)
pdb4an9.ent
RDF4an9.rdf.gz Visualize(78.79 KB)
4an9.rdf
Structure factorsr4an9sf.ent.gz Display(114.03 KB)
r4an9sf.ent
Biological unit (mmCIF format)4an9-assembly1.cif.gz Display(60.33 KB)
4an9-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)4an9.pdb1.gz Display(46.29 KB)
4an9.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF4an9_validation.pdf.gz Display(1006.07 KB)
4an9_validation.pdf
PDF-full4an9_full_validation.pdf.gz Display(1015.72 KB)
4an9_full_validation.pdf
mmCIF4an9_validation.cif.gz Display(18.12 KB)
4an9_validation.cif
XML4an9_validation.xml.gz Display(13.94 KB)
4an9_validation.xml
PNG4an9_multipercentile_validation.png.gz Display(166.43 KB)
4an9_multipercentile_validation.png
SVG4an9_multipercentile_validation.svg.gz Display(976.00 B)
4an9_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)4an9_validation_2fo-fc_map_coef.cif.gz Display(83.47 KB)
4an9_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)4an9_validation_fo-fc_map_coef.cif.gz Display(81.83 KB)
4an9_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)4an9_validation_2fo-fc_map_coef.mtz Visualize(199.64 KB)
fo-fc (MTZ)4an9_validation_fo-fc_map_coef.mtz Visualize(199.64 KB)

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PDB entries from 2024-07-17

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