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4AN3

Crystal structures of human MEK1 with carboxamide-based allosteric inhibitor XL518 (GDC-0973), or related analogs.

Resources
File formatFile name (file size)
PDBx/mmCIF4an3.cif.gz Display(74.17 KB)
4an3.cif
PDBx/mmJSONall4an3.json.gz Display (Tree)(51.50 KB)
4an3.json
no-atom4an3-noatom.json.gz Display (Header)(14.31 KB)
4an3-noatom.json
add only4an3-plus.json.gz Display(1.27 KB)
4an3-plus.json
PDBMLall4an3.xml.gz Display(98.11 KB)
4an3.xml
no-atom4an3-noatom.xml.gz Display(27.52 KB)
4an3-noatom.xml
ext-atom4an3-extatom.xml.gz Display(52.94 KB)
4an3-extatom.xml
PDBpdb4an3.ent.gz Display(53.72 KB)
pdb4an3.ent
RDF4an3.rdf.gz Visualize(79.70 KB)
4an3.rdf
Structure factorsr4an3sf.ent.gz Display(264.40 KB)
r4an3sf.ent
Biological unit (mmCIF format)4an3-assembly1.cif.gz Display(62.74 KB)
4an3-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)4an3.pdb1.gz Display(48.09 KB)
4an3.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF4an3_validation.pdf.gz Display(1.01 MB)
4an3_validation.pdf
PDF-full4an3_full_validation.pdf.gz Display(1.02 MB)
4an3_full_validation.pdf
mmCIF4an3_validation.cif.gz Display(19.87 KB)
4an3_validation.cif
XML4an3_validation.xml.gz Display(14.74 KB)
4an3_validation.xml
PNG4an3_multipercentile_validation.png.gz Display(168.66 KB)
4an3_multipercentile_validation.png
SVG4an3_multipercentile_validation.svg.gz Display(974.00 B)
4an3_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)4an3_validation_2fo-fc_map_coef.cif.gz Display(197.80 KB)
4an3_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)4an3_validation_fo-fc_map_coef.cif.gz Display(194.04 KB)
4an3_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)4an3_validation_2fo-fc_map_coef.mtz Visualize(469.69 KB)
fo-fc (MTZ)4an3_validation_fo-fc_map_coef.mtz Visualize(469.69 KB)

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PDB entries from 2024-08-21

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