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4AGW

Discovery of a small molecule type II inhibitor of wild-type and gatekeeper mutants of BCR-ABL, PDGFRalpha, Kit, and Src kinases

Resources
File formatFile name (file size)
PDBx/mmCIF4agw.cif.gz Display(123.89 KB)
4agw.cif
PDBx/mmJSONall4agw.json.gz Display (Tree)(81.35 KB)
4agw.json
no-atom4agw-noatom.json.gz Display (Header)(15.49 KB)
4agw-noatom.json
add only4agw-plus.json.gz Display(1.11 KB)
4agw-plus.json
PDBMLall4agw.xml.gz Display(168.14 KB)
4agw.xml
no-atom4agw-noatom.xml.gz Display(34.26 KB)
4agw-noatom.xml
ext-atom4agw-extatom.xml.gz Display(100.39 KB)
4agw-extatom.xml
PDBpdb4agw.ent.gz Display(96.25 KB)
pdb4agw.ent
RDF4agw.rdf.gz Visualize(99.40 KB)
4agw.rdf
Structure factorsr4agwsf.ent.gz Display(259.46 KB)
r4agwsf.ent
Biological unit (mmCIF format)4agw-assembly1.cif.gz Display(59.90 KB)
4agw-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

4agw-assembly2.cif.gz Display(59.59 KB)
4agw-assembly2.cif (B)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)4agw.pdb1.gz Display(46.46 KB)
4agw.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

4agw.pdb2.gz Display(46.73 KB)
4agw.pdb2 (B)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF4agw_validation.pdf.gz Display(842.09 KB)
4agw_validation.pdf
PDF-full4agw_full_validation.pdf.gz Display(889.06 KB)
4agw_full_validation.pdf
mmCIF4agw_validation.cif.gz Display(40.62 KB)
4agw_validation.cif
XML4agw_validation.xml.gz Display(31.30 KB)
4agw_validation.xml
PNG4agw_multipercentile_validation.png.gz Display(173.26 KB)
4agw_multipercentile_validation.png
SVG4agw_multipercentile_validation.svg.gz Display(977.00 B)
4agw_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)4agw_validation_2fo-fc_map_coef.cif.gz Display(408.44 KB)
4agw_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)4agw_validation_fo-fc_map_coef.cif.gz Display(369.41 KB)
4agw_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)4agw_validation_2fo-fc_map_coef.mtz Visualize(663.90 KB)
fo-fc (MTZ)4agw_validation_fo-fc_map_coef.mtz Visualize(663.90 KB)

222926

PDB entries from 2024-07-24

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