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3SFI

Ethionamide Boosters Part 2: Combining Bioisosteric Replacement and Structure-Based Drug Design to Solve Pharmacokinetic Issues in a Series of Potent 1,2,4-Oxadiazole EthR Inhibitors.

Resources
File formatFile name (file size)
PDBx/mmCIF3sfi.cif.gz Display(52.48 KB)
3sfi.cif
PDBx/mmJSONall3sfi.json.gz Display (Tree)(36.66 KB)
3sfi.json
no-atom3sfi-noatom.json.gz Display (Header)(10.71 KB)
3sfi-noatom.json
add only3sfi-plus.json.gz Display(954.00 B)
3sfi-plus.json
PDBMLall3sfi.xml.gz Display(67.66 KB)
3sfi.xml
no-atom3sfi-noatom.xml.gz Display(21.44 KB)
3sfi-noatom.xml
ext-atom3sfi-extatom.xml.gz Display(34.55 KB)
3sfi-extatom.xml
PDBpdb3sfi.ent.gz Display(36.53 KB)
pdb3sfi.ent
RDF3sfi.rdf.gz Visualize(64.57 KB)
3sfi.rdf
Structure factorsr3sfisf.ent.gz Display(168.93 KB)
r3sfisf.ent
Biological unit (mmCIF format)3sfi-assembly1.cif.gz Display(77.55 KB)
3sfi-assembly1.cif (A)

*author and software defined assembly, 2 molecule(s) (dimeric)

Biological unit (PDB format)3sfi.pdb1.gz Display(61.27 KB)
3sfi.pdb1 (A)

*author and software defined assembly, 2 molecule(s) (dimeric)

Validation reportsPDF3sfi_validation.pdf.gz Display(675.40 KB)
3sfi_validation.pdf
PDF-full3sfi_full_validation.pdf.gz Display(676.91 KB)
3sfi_full_validation.pdf
mmCIF3sfi_validation.cif.gz Display(12.10 KB)
3sfi_validation.cif
XML3sfi_validation.xml.gz Display(9.53 KB)
3sfi_validation.xml
PNG3sfi_multipercentile_validation.png.gz Display(170.69 KB)
3sfi_multipercentile_validation.png
SVG3sfi_multipercentile_validation.svg.gz Display(957.00 B)
3sfi_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)3sfi_validation_2fo-fc_map_coef.cif.gz Display(110.51 KB)
3sfi_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)3sfi_validation_fo-fc_map_coef.cif.gz Display(108.63 KB)
3sfi_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)3sfi_validation_2fo-fc_map_coef.mtz Visualize(271.40 KB)
fo-fc (MTZ)3sfi_validation_fo-fc_map_coef.mtz Visualize(271.40 KB)

222926

PDB entries from 2024-07-24

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