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3RKZ

Discovery of a stable macrocyclic o-aminobenzamide Hsp90 inhibitor capable of significantly decreasing tumor volume in a mouse xenograft model.

Resources
File formatFile name (file size)
PDBx/mmCIF3rkz.cif.gz Display(64.99 KB)
3rkz.cif
PDBx/mmJSONall3rkz.json.gz Display (Tree)(46.46 KB)
3rkz.json
no-atom3rkz-noatom.json.gz Display (Header)(13.01 KB)
3rkz-noatom.json
add only3rkz-plus.json.gz Display(1.22 KB)
3rkz-plus.json
PDBMLall3rkz.xml.gz Display(86.39 KB)
3rkz.xml
no-atom3rkz-noatom.xml.gz Display(26.18 KB)
3rkz-noatom.xml
ext-atom3rkz-extatom.xml.gz Display(44.70 KB)
3rkz-extatom.xml
PDBpdb3rkz.ent.gz Display(46.06 KB)
pdb3rkz.ent
RDF3rkz.rdf.gz Visualize(73.28 KB)
3rkz.rdf
Structure factorsr3rkzsf.ent.gz Display(570.79 KB)
r3rkzsf.ent
Biological unit (mmCIF format)3rkz-assembly1.cif.gz Display(54.16 KB)
3rkz-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)3rkz.pdb1.gz Display(40.81 KB)
3rkz.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF3rkz_validation.pdf.gz Display(843.08 KB)
3rkz_validation.pdf
PDF-full3rkz_full_validation.pdf.gz Display(844.17 KB)
3rkz_full_validation.pdf
mmCIF3rkz_validation.cif.gz Display(21.06 KB)
3rkz_validation.cif
XML3rkz_validation.xml.gz Display(13.75 KB)
3rkz_validation.xml
PNG3rkz_multipercentile_validation.png.gz Display(160.79 KB)
3rkz_multipercentile_validation.png
SVG3rkz_multipercentile_validation.svg.gz Display(953.00 B)
3rkz_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)3rkz_validation_2fo-fc_map_coef.cif.gz Display(407.95 KB)
3rkz_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)3rkz_validation_fo-fc_map_coef.cif.gz Display(363.56 KB)
3rkz_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)3rkz_validation_2fo-fc_map_coef.mtz Visualize(983.66 KB)
fo-fc (MTZ)3rkz_validation_fo-fc_map_coef.mtz Visualize(983.66 KB)

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PDB entries from 2024-07-17

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