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3R22

Design, synthesis, and biological evaluation of pyrazolopyridine-sulfonamides as potent multiple-mitotic kinase (MMK) inhibitors (Part I)

Resources
File formatFile name (file size)
PDBx/mmCIF3r22.cif.gz Display(66.67 KB)
3r22.cif
PDBx/mmJSONall3r22.json.gz Display (Tree)(46.95 KB)
3r22.json
no-atom3r22-noatom.json.gz Display (Header)(12.27 KB)
3r22-noatom.json
add only3r22-plus.json.gz Display(1.44 KB)
3r22-plus.json
PDBMLall3r22.xml.gz Display(87.27 KB)
3r22.xml
no-atom3r22-noatom.xml.gz Display(24.87 KB)
3r22-noatom.xml
ext-atom3r22-extatom.xml.gz Display(46.88 KB)
3r22-extatom.xml
PDBpdb3r22.ent.gz Display(48.14 KB)
pdb3r22.ent
RDF3r22.rdf.gz Visualize(73.47 KB)
3r22.rdf
Structure factorsr3r22sf.ent.gz Display(115.50 KB)
r3r22sf.ent
Biological unit (mmCIF format)3r22-assembly1.cif.gz Display(55.03 KB)
3r22-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)3r22.pdb1.gz Display(42.54 KB)
3r22.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF3r22_validation.pdf.gz Display(734.52 KB)
3r22_validation.pdf
PDF-full3r22_full_validation.pdf.gz Display(744.40 KB)
3r22_full_validation.pdf
mmCIF3r22_validation.cif.gz Display(16.90 KB)
3r22_validation.cif
XML3r22_validation.xml.gz Display(13.09 KB)
3r22_validation.xml
PNG3r22_multipercentile_validation.png.gz Display(167.99 KB)
3r22_multipercentile_validation.png
SVG3r22_multipercentile_validation.svg.gz Display(978.00 B)
3r22_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)3r22_validation_2fo-fc_map_coef.cif.gz Display(76.07 KB)
3r22_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)3r22_validation_fo-fc_map_coef.cif.gz Display(74.73 KB)
3r22_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)3r22_validation_2fo-fc_map_coef.mtz Visualize(185.74 KB)
fo-fc (MTZ)3r22_validation_fo-fc_map_coef.mtz Visualize(185.74 KB)

222036

PDB entries from 2024-07-03

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