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3R21

Design, synthesis, and biological evaluation of pyrazolopyridine-sulfonamides as potent multiple-mitotic kinase (MMK) inhibitors (Part I)

Resources
File formatFile name (file size)
PDBx/mmCIF3r21.cif.gz Display(67.54 KB)
3r21.cif
PDBx/mmJSONall3r21.json.gz Display (Tree)(47.17 KB)
3r21.json
no-atom3r21-noatom.json.gz Display (Header)(12.27 KB)
3r21-noatom.json
add only3r21-plus.json.gz Display(1.43 KB)
3r21-plus.json
PDBMLall3r21.xml.gz Display(88.24 KB)
3r21.xml
no-atom3r21-noatom.xml.gz Display(24.27 KB)
3r21-noatom.xml
ext-atom3r21-extatom.xml.gz Display(47.75 KB)
3r21-extatom.xml
PDBpdb3r21.ent.gz Display(49.29 KB)
pdb3r21.ent
RDF3r21.rdf.gz Visualize(72.08 KB)
3r21.rdf
Structure factorsr3r21sf.ent.gz Display(116.77 KB)
r3r21sf.ent
Biological unit (mmCIF format)3r21-assembly1.cif.gz Display(56.22 KB)
3r21-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)3r21.pdb1.gz Display(43.42 KB)
3r21.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF3r21_validation.pdf.gz Display(753.26 KB)
3r21_validation.pdf
PDF-full3r21_full_validation.pdf.gz Display(763.58 KB)
3r21_full_validation.pdf
mmCIF3r21_validation.cif.gz Display(16.69 KB)
3r21_validation.cif
XML3r21_validation.xml.gz Display(13.11 KB)
3r21_validation.xml
PNG3r21_multipercentile_validation.png.gz Display(165.73 KB)
3r21_multipercentile_validation.png
SVG3r21_multipercentile_validation.svg.gz Display(976.00 B)
3r21_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)3r21_validation_2fo-fc_map_coef.cif.gz Display(76.72 KB)
3r21_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)3r21_validation_fo-fc_map_coef.cif.gz Display(75.17 KB)
3r21_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)3r21_validation_2fo-fc_map_coef.mtz Visualize(187.64 KB)
fo-fc (MTZ)3r21_validation_fo-fc_map_coef.mtz Visualize(187.64 KB)

219140

PDB entries from 2024-05-01

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