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3PRE

Quinazolines with intra-molecular hydrogen bonding scaffold (iMHBS) as PI3K/mTOR dual inhibitors.

Resources
File formatFile name (file size)
PDBx/mmCIF3pre.cif.gz Display(183.83 KB)
3pre.cif
PDBx/mmJSONall3pre.json.gz Display (Tree)(121.16 KB)
3pre.json
no-atom3pre-noatom.json.gz Display (Header)(20.79 KB)
3pre-noatom.json
add only3pre-plus.json.gz Display(1.00 KB)
3pre-plus.json
PDBMLall3pre.xml.gz Display(244.22 KB)
3pre.xml
no-atom3pre-noatom.xml.gz Display(42.58 KB)
3pre-noatom.xml
ext-atom3pre-extatom.xml.gz Display(152.37 KB)
3pre-extatom.xml
PDBpdb3pre.ent.gz Display(141.86 KB)
pdb3pre.ent
RDF3pre.rdf.gz Visualize(131.21 KB)
3pre.rdf
Structure factorsr3presf.ent.gz Display(317.37 KB)
r3presf.ent
Biological unit (mmCIF format)3pre-assembly1.cif.gz Display(172.66 KB)
3pre-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)3pre.pdb1.gz Display(135.66 KB)
3pre.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF3pre_validation.pdf.gz Display(728.99 KB)
3pre_validation.pdf
PDF-full3pre_full_validation.pdf.gz Display(759.55 KB)
3pre_full_validation.pdf
mmCIF3pre_validation.cif.gz Display(44.33 KB)
3pre_validation.cif
XML3pre_validation.xml.gz Display(32.75 KB)
3pre_validation.xml
PNG3pre_multipercentile_validation.png.gz Display(167.02 KB)
3pre_multipercentile_validation.png
SVG3pre_multipercentile_validation.svg.gz Display(978.00 B)
3pre_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)3pre_validation_2fo-fc_map_coef.cif.gz Display(231.50 KB)
3pre_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)3pre_validation_fo-fc_map_coef.cif.gz Display(226.40 KB)
3pre_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)3pre_validation_2fo-fc_map_coef.mtz Visualize(531.38 KB)
fo-fc (MTZ)3pre_validation_fo-fc_map_coef.mtz Visualize(531.38 KB)

221051

PDB entries from 2024-06-12

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