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3L16

Discovery of (thienopyrimidin-2-yl)aminopyrimidines as Potent, Selective, and Orally Available Pan-PI3-Kinase and Dual Pan-PI3-Kinase/mTOR Inhibitors for the Treatment of Cancer

Resources
File formatFile name (file size)
PDBx/mmCIF3l16.cif.gz Display(186.42 KB)
3l16.cif
PDBx/mmJSONall3l16.json.gz Display (Tree)(127.54 KB)
3l16.json
no-atom3l16-noatom.json.gz Display (Header)(24.03 KB)
3l16-noatom.json
add only3l16-plus.json.gz Display(1.10 KB)
3l16-plus.json
PDBMLall3l16.xml.gz Display(249.22 KB)
3l16.xml
no-atom3l16-noatom.xml.gz Display(43.77 KB)
3l16-noatom.xml
ext-atom3l16-extatom.xml.gz Display(154.38 KB)
3l16-extatom.xml
PDBpdb3l16.ent.gz Display(144.04 KB)
pdb3l16.ent
RDF3l16.rdf.gz Visualize(133.17 KB)
3l16.rdf
Structure factorsr3l16sf.ent.gz Display(338.48 KB)
r3l16sf.ent
Biological unit (mmCIF format)3l16-assembly1.cif.gz Display(174.32 KB)
3l16-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)3l16.pdb1.gz Display(137.53 KB)
3l16.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF3l16_validation.pdf.gz Display(878.04 KB)
3l16_validation.pdf
PDF-full3l16_full_validation.pdf.gz Display(899.94 KB)
3l16_full_validation.pdf
mmCIF3l16_validation.cif.gz Display(42.08 KB)
3l16_validation.cif
XML3l16_validation.xml.gz Display(30.85 KB)
3l16_validation.xml
PNG3l16_multipercentile_validation.png.gz Display(165.12 KB)
3l16_multipercentile_validation.png
SVG3l16_multipercentile_validation.svg.gz Display(973.00 B)
3l16_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)3l16_validation_2fo-fc_map_coef.cif.gz Display(229.59 KB)
3l16_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)3l16_validation_fo-fc_map_coef.cif.gz Display(224.59 KB)
3l16_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)3l16_validation_2fo-fc_map_coef.mtz Visualize(530.87 KB)
fo-fc (MTZ)3l16_validation_fo-fc_map_coef.mtz Visualize(530.87 KB)

222926

PDB entries from 2024-07-24

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