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3K5K

Discovery of a 2,4-Diamino-7-aminoalkoxy-quinazoline as a Potent Inhibitor of Histone Lysine Methyltransferase, G9a

Resources
File formatFile name (file size)
PDBx/mmCIF3k5k.cif.gz Display(137.90 KB)
3k5k.cif
PDBx/mmJSONall3k5k.json.gz Display (Tree)(90.56 KB)
3k5k.json
no-atom3k5k-noatom.json.gz Display (Header)(19.66 KB)
3k5k-noatom.json
add only3k5k-plus.json.gz Display(1.45 KB)
3k5k-plus.json
PDBMLall3k5k.xml.gz Display(187.16 KB)
3k5k.xml
no-atom3k5k-noatom.xml.gz Display(43.50 KB)
3k5k-noatom.xml
ext-atom3k5k-extatom.xml.gz Display(107.91 KB)
3k5k-extatom.xml
pdb_nextgenallpdb_00003k5k_xyz-enrich.cif.gz Display(154.23 KB)
pdb_00003k5k_xyz-enrich.cif
no-atompdb_00003k5k_xyz-no-atom-enrich.xml.gz Display(60.35 KB)
pdb_00003k5k_xyz-no-atom-enrich.xml
ng-only3k5k-plus.json.gz Display(3.61 KB)
3k5k-plus.json
PDBpdb3k5k.ent.gz Display(103.94 KB)
pdb3k5k.ent
RDF3k5k.rdf.gz Visualize(117.45 KB)
3k5k.rdf
Structure factorsr3k5ksf.ent.gz Display(999.85 KB)
r3k5ksf.ent
Biological unit (mmCIF format)3k5k-assembly1.cif.gz Display(65.34 KB)
3k5k-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

3k5k-assembly2.cif.gz Display(64.32 KB)
3k5k-assembly2.cif (B)

*author defined assembly, 1 molecule(s) (monomeric)

3k5k-assembly3.cif.gz Display(122.70 KB)
3k5k-assembly3.cif (A,B)

*software defined assembly, 2 molecule(s) (dimeric)

Biological unit (PDB format)3k5k.pdb1.gz Display(51.06 KB)
3k5k.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

3k5k.pdb2.gz Display(49.66 KB)
3k5k.pdb2 (B)

*author defined assembly, 1 molecule(s) (monomeric)

3k5k.pdb3.gz Display(96.91 KB)
3k5k.pdb3 (A,B)

*software defined assembly, 2 molecule(s) (dimeric)

Validation reportsPDF3k5k_validation.pdf.gz Display(1.54 MB)
3k5k_validation.pdf
PDF-full3k5k_full_validation.pdf.gz Display(1.54 MB)
3k5k_full_validation.pdf
mmCIF3k5k_validation.cif.gz Display(22.42 KB)
3k5k_validation.cif
XML3k5k_validation.xml.gz Display(13.98 KB)
3k5k_validation.xml
PNG3k5k_multipercentile_validation.png.gz Display(124.95 KB)
3k5k_multipercentile_validation.png
SVG3k5k_multipercentile_validation.svg.gz Display(803.00 B)
3k5k_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)3k5k_validation_2fo-fc_map_coef.cif.gz Display(1.00 MB)
3k5k_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)3k5k_validation_fo-fc_map_coef.cif.gz Display(1.00 MB)
3k5k_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)3k5k_validation_2fo-fc_map_coef.mtz Visualize(1.59 MB)
fo-fc (MTZ)3k5k_validation_fo-fc_map_coef.mtz Visualize(1.59 MB)

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PDB entries from 2025-06-18

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