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3JYA

Discovery of 3H-benzo[4,5]thieno[3,2-d]pyrimidin-4-ones as Potent, Highly Selective and Orally Bioavailable Pim Kinases Inhibitors

Resources
File formatFile name (file size)
PDBx/mmCIF3jya.cif.gz Display(68.31 KB)
3jya.cif
PDBx/mmJSONall3jya.json.gz Display (Tree)(47.15 KB)
3jya.json
no-atom3jya-noatom.json.gz Display (Header)(11.80 KB)
3jya-noatom.json
add only3jya-plus.json.gz Display(2.03 KB)
3jya-plus.json
PDBMLall3jya.xml.gz Display(89.57 KB)
3jya.xml
no-atom3jya-noatom.xml.gz Display(22.24 KB)
3jya-noatom.xml
ext-atom3jya-extatom.xml.gz Display(50.64 KB)
3jya-extatom.xml
PDBpdb3jya.ent.gz Display(50.23 KB)
pdb3jya.ent
RDF3jya.rdf.gz Visualize(67.76 KB)
3jya.rdf
Structure factorsr3jyasf.ent.gz Display(374.15 KB)
r3jyasf.ent
Biological unit (mmCIF format)3jya-assembly1.cif.gz Display(59.23 KB)
3jya-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)3jya.pdb1.gz Display(45.66 KB)
3jya.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF3jya_validation.pdf.gz Display(804.17 KB)
3jya_validation.pdf
PDF-full3jya_full_validation.pdf.gz Display(807.27 KB)
3jya_full_validation.pdf
mmCIF3jya_validation.cif.gz Display(15.33 KB)
3jya_validation.cif
XML3jya_validation.xml.gz Display(12.04 KB)
3jya_validation.xml
PNG3jya_multipercentile_validation.png.gz Display(171.57 KB)
3jya_multipercentile_validation.png
SVG3jya_multipercentile_validation.svg.gz Display(980.00 B)
3jya_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)3jya_validation_2fo-fc_map_coef.cif.gz Display(250.98 KB)
3jya_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)3jya_validation_fo-fc_map_coef.cif.gz Display(238.90 KB)
3jya_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)3jya_validation_2fo-fc_map_coef.mtz Visualize(593.86 KB)
fo-fc (MTZ)3jya_validation_fo-fc_map_coef.mtz Visualize(593.86 KB)

222926

PDB entries from 2024-07-24

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