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3JY0

Discovery of 3H-benzo[4,5]thieno[3,2-d]pyrimidin-4-ones as Potent, Highly Selective and Orally Bioavailable Pim Kinases Inhibitors

Resources
File formatFile name (file size)
PDBx/mmCIF3jy0.cif.gz Display(68.88 KB)
3jy0.cif
PDBx/mmJSONall3jy0.json.gz Display (Tree)(47.98 KB)
3jy0.json
no-atom3jy0-noatom.json.gz Display (Header)(12.30 KB)
3jy0-noatom.json
add only3jy0-plus.json.gz Display(2.03 KB)
3jy0-plus.json
PDBMLall3jy0.xml.gz Display(91.23 KB)
3jy0.xml
no-atom3jy0-noatom.xml.gz Display(22.99 KB)
3jy0-noatom.xml
ext-atom3jy0-extatom.xml.gz Display(50.79 KB)
3jy0-extatom.xml
PDBpdb3jy0.ent.gz Display(50.48 KB)
pdb3jy0.ent
RDF3jy0.rdf.gz Visualize(69.77 KB)
3jy0.rdf
Structure factorsr3jy0sf.ent.gz Display(262.60 KB)
r3jy0sf.ent
Biological unit (mmCIF format)3jy0-assembly1.cif.gz Display(59.26 KB)
3jy0-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)3jy0.pdb1.gz Display(45.69 KB)
3jy0.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF3jy0_validation.pdf.gz Display(763.06 KB)
3jy0_validation.pdf
PDF-full3jy0_full_validation.pdf.gz Display(770.86 KB)
3jy0_full_validation.pdf
mmCIF3jy0_validation.cif.gz Display(16.97 KB)
3jy0_validation.cif
XML3jy0_validation.xml.gz Display(13.27 KB)
3jy0_validation.xml
PNG3jy0_multipercentile_validation.png.gz Display(165.83 KB)
3jy0_multipercentile_validation.png
SVG3jy0_multipercentile_validation.svg.gz Display(975.00 B)
3jy0_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)3jy0_validation_2fo-fc_map_coef.cif.gz Display(174.63 KB)
3jy0_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)3jy0_validation_fo-fc_map_coef.cif.gz Display(171.59 KB)
3jy0_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)3jy0_validation_2fo-fc_map_coef.mtz Visualize(411.12 KB)
fo-fc (MTZ)3jy0_validation_fo-fc_map_coef.mtz Visualize(411.12 KB)

222036

PDB entries from 2024-07-03

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