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3EY4

Further studies with the 2-amino-1,3-thiazol-4(5H)-one class of 11-hydroxysteroid dehydrogenase type 1 (11-HSD1) inhibitors: Reducing pregnane X receptor (PXR) activity and exploring activity in a monkey pharmacodynamic model

Resources
File formatFile name (file size)
PDBx/mmCIF3ey4.cif.gz Display(211.07 KB)
3ey4.cif
PDBx/mmJSONall3ey4.json.gz Display (Tree)(131.63 KB)
3ey4.json
no-atom3ey4-noatom.json.gz Display (Header)(16.55 KB)
3ey4-noatom.json
add only3ey4-plus.json.gz Display(1.94 KB)
3ey4-plus.json
PDBMLall3ey4.xml.gz Display(287.46 KB)
3ey4.xml
no-atom3ey4-noatom.xml.gz Display(44.04 KB)
3ey4-noatom.xml
ext-atom3ey4-extatom.xml.gz Display(184.81 KB)
3ey4-extatom.xml
PDBpdb3ey4.ent.gz Display(170.98 KB)
pdb3ey4.ent
RDF3ey4.rdf.gz Visualize(126.43 KB)
3ey4.rdf
Structure factorsr3ey4sf.ent.gz Display(341.13 KB)
r3ey4sf.ent
Biological unit (mmCIF format)3ey4-assembly1.cif.gz Display(102.38 KB)
3ey4-assembly1.cif (A,B)

*author and software defined assembly, 2 molecule(s) (dimeric)

3ey4-assembly2.cif.gz Display(103.72 KB)
3ey4-assembly2.cif (C,D)

*author and software defined assembly, 2 molecule(s) (dimeric)

Biological unit (PDB format)3ey4.pdb1.gz Display(83.82 KB)
3ey4.pdb1 (A,B)

*author and software defined assembly, 2 molecule(s) (dimeric)

3ey4.pdb2.gz Display(84.21 KB)
3ey4.pdb2 (C,D)

*author and software defined assembly, 2 molecule(s) (dimeric)

Validation reportsPDF3ey4_validation.pdf.gz Display(2.38 MB)
3ey4_validation.pdf
PDF-full3ey4_full_validation.pdf.gz Display(2.43 MB)
3ey4_full_validation.pdf
mmCIF3ey4_validation.cif.gz Display(59.58 KB)
3ey4_validation.cif
XML3ey4_validation.xml.gz Display(46.51 KB)
3ey4_validation.xml
PNG3ey4_multipercentile_validation.png.gz Display(169.15 KB)
3ey4_multipercentile_validation.png
SVG3ey4_multipercentile_validation.svg.gz Display(980.00 B)
3ey4_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)3ey4_validation_2fo-fc_map_coef.cif.gz Display(256.06 KB)
3ey4_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)3ey4_validation_fo-fc_map_coef.cif.gz Display(245.05 KB)
3ey4_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)3ey4_validation_2fo-fc_map_coef.mtz Visualize(604.70 KB)
fo-fc (MTZ)3ey4_validation_fo-fc_map_coef.mtz Visualize(604.70 KB)

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PDB entries from 2024-07-10

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