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2WPA

Optimisation of 6,6-Dimethyl Pyrrolo 3,4-c pyrazoles: Identification of PHA-793887, a Potent CDK Inhibitor Suitable for Intravenous Dosing

Resources
File formatFile name (file size)
PDBx/mmCIF2wpa.cif.gz Display(238.63 KB)
2wpa.cif
PDBx/mmJSONall2wpa.json.gz Display (Tree)(154.67 KB)
2wpa.json
no-atom2wpa-noatom.json.gz Display (Header)(19.15 KB)
2wpa-noatom.json
add only2wpa-plus.json.gz Display(2.77 KB)
2wpa-plus.json
PDBMLall2wpa.xml.gz Display(324.84 KB)
2wpa.xml
no-atom2wpa-noatom.xml.gz Display(48.45 KB)
2wpa-noatom.xml
ext-atom2wpa-extatom.xml.gz Display(210.02 KB)
2wpa-extatom.xml
PDBpdb2wpa.ent.gz Display(194.05 KB)
pdb2wpa.ent
RDF2wpa.rdf.gz Visualize(137.82 KB)
2wpa.rdf
Structure factorsr2wpasf.ent.gz Display(596.16 KB)
r2wpasf.ent
Biological unit (mmCIF format)2wpa-assembly1.cif.gz Display(118.80 KB)
2wpa-assembly1.cif (A,B)

*author and software defined assembly, 2 molecule(s) (dimeric)

2wpa-assembly2.cif.gz Display(118.00 KB)
2wpa-assembly2.cif (C,D)

*author and software defined assembly, 2 molecule(s) (dimeric)

Biological unit (PDB format)2wpa.pdb1.gz Display(94.63 KB)
2wpa.pdb1 (A,B)

*author and software defined assembly, 2 molecule(s) (dimeric)

2wpa.pdb2.gz Display(94.20 KB)
2wpa.pdb2 (C,D)

*author and software defined assembly, 2 molecule(s) (dimeric)

Validation reportsPDF2wpa_validation.pdf.gz Display(1.05 MB)
2wpa_validation.pdf
PDF-full2wpa_full_validation.pdf.gz Display(1.07 MB)
2wpa_full_validation.pdf
mmCIF2wpa_validation.cif.gz Display(61.51 KB)
2wpa_validation.cif
XML2wpa_validation.xml.gz Display(43.94 KB)
2wpa_validation.xml
PNG2wpa_multipercentile_validation.png.gz Display(168.88 KB)
2wpa_multipercentile_validation.png
SVG2wpa_multipercentile_validation.svg.gz Display(977.00 B)
2wpa_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)2wpa_validation_2fo-fc_map_coef.cif.gz Display(765.56 KB)
2wpa_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)2wpa_validation_fo-fc_map_coef.cif.gz Display(749.63 KB)
2wpa_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)2wpa_validation_2fo-fc_map_coef.mtz Visualize(1.74 MB)
fo-fc (MTZ)2wpa_validation_fo-fc_map_coef.mtz Visualize(1.74 MB)

224004

PDB entries from 2024-08-21

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