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1EAS

NONPEPTIDIC INHIBITORS OF HUMAN LEUKOCYTE ELASTASE. 3. DESIGN, SYNTHESIS, X-RAY CRYSTALLOGRAPHIC ANALYSIS, AND STRUCTURE-ACTIVITY RELATIONSHIPS FOR A SERIES OF ORALLY ACTIVE 3-AMINO-6-PHENYLPYRIDIN-2-ONE TRIFLUOROMETHYL KETONES

Resources
File formatFile name (file size)
PDBx/mmCIF1eas.cif.gz Display(65.22 KB)
1eas.cif
PDBx/mmJSONall1eas.json.gz Display (Tree)(45.84 KB)
1eas.json
no-atom1eas-noatom.json.gz Display (Header)(14.10 KB)
1eas-noatom.json
add only1eas-plus.json.gz Display(1.77 KB)
1eas-plus.json
PDBMLall1eas.xml.gz Display(87.17 KB)
1eas.xml
no-atom1eas-noatom.xml.gz Display(26.00 KB)
1eas-noatom.xml
ext-atom1eas-extatom.xml.gz Display(45.15 KB)
1eas-extatom.xml
pdb_nextgenallpdb_00001eas_xyz-enrich.cif.gz Display(72.84 KB)
pdb_00001eas_xyz-enrich.cif
no-atompdb_00001eas_xyz-no-atom-enrich.xml.gz Display(35.05 KB)
pdb_00001eas_xyz-no-atom-enrich.xml
ng-only1eas-plus.json.gz Display(2.17 KB)
1eas-plus.json
PDBpdb1eas.ent.gz Display(46.20 KB)
pdb1eas.ent
RDF1eas.rdf.gz Visualize(74.90 KB)
1eas.rdf
Structure factorsr1eassf.ent.gz Display(136.87 KB)
r1eassf.ent
Biological unit (mmCIF format)1eas-assembly1.cif.gz Display(55.01 KB)
1eas-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)1eas.pdb1.gz Display(42.20 KB)
1eas.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF1eas_validation.pdf.gz Display(768.97 KB)
1eas_validation.pdf
PDF-full1eas_full_validation.pdf.gz Display(771.11 KB)
1eas_full_validation.pdf
mmCIF1eas_validation.cif.gz Display(17.36 KB)
1eas_validation.cif
XML1eas_validation.xml.gz Display(12.61 KB)
1eas_validation.xml
PNG1eas_multipercentile_validation.png.gz Display(153.68 KB)
1eas_multipercentile_validation.png
SVG1eas_multipercentile_validation.svg.gz Display(903.00 B)
1eas_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)1eas_validation_2fo-fc_map_coef.cif.gz Display(303.77 KB)
1eas_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)1eas_validation_fo-fc_map_coef.cif.gz Display(287.67 KB)
1eas_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)1eas_validation_2fo-fc_map_coef.mtz Visualize(512.66 KB)
fo-fc (MTZ)1eas_validation_fo-fc_map_coef.mtz Visualize(512.66 KB)

238268

PDB entries from 2025-07-02

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