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10MV

N-Alkyl & N-Aryl Aminopyrazole Spirocarbamates: A Two-Pronged Lead Optimization Strategy to Identify Orally Bioavailable Plasma Kallikrein Inhibitors complex with Compound 15 ((3'R)-1'-(5-amino-1-phenyl-1H-pyrazole-4-carbonyl)-6-chloro-5-fluorospiro[[3,1]benzoxazine-4,3'-piperidin]-2(1H)-one)

This is a non-PDB format compatible entry.
Resources
File formatFile name (file size)
PDBx/mmCIF10mv.cif.gz Display(206.86 KB)
10mv.cif
PDBx/mmJSONall10mv.json.gz Display (Tree)(139.43 KB)
10mv.json
no-atom10mv-noatom.json.gz Display (Header)(16.34 KB)
10mv-noatom.json
add only10mv-plus.json.gz Display(724.00 B)
10mv-plus.json
PDBMLall10mv.xml.gz Display(271.14 KB)
10mv.xml
no-atom10mv-noatom.xml.gz Display(26.58 KB)
10mv-noatom.xml
ext-atom10mv-extatom.xml.gz Display(93.99 KB)
10mv-extatom.xml
pdb_nextgenallpdb_000010mv_xyz-enrich.cif.gz Display(213.99 KB)
pdb_000010mv_xyz-enrich.cif
no-atompdb_000010mv_xyz-no-atom-enrich.xml.gz Display(30.36 KB)
pdb_000010mv_xyz-no-atom-enrich.xml
ng-only10mv-plus.json.gz Display(2.30 KB)
10mv-plus.json
RDF10mv.rdf.gz Visualize(78.04 KB)
10mv.rdf
Structure factorsr10mvsf.ent.gz Display(1.69 MB)
r10mvsf.ent
Biological unit (mmCIF format)10mv-assembly1.cif.gz Display(196.18 KB)
10mv-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF10mv_validation.pdf.gz Display(759.11 KB)
10mv_validation.pdf
PDF-full10mv_full_validation.pdf.gz Display(763.35 KB)
10mv_full_validation.pdf
mmCIF10mv_validation.cif.gz Display(19.02 KB)
10mv_validation.cif
XML10mv_validation.xml.gz Display(13.89 KB)
10mv_validation.xml
PNG10mv_multipercentile_validation.png.gz Display(158.45 KB)
10mv_multipercentile_validation.png
SVG10mv_multipercentile_validation.svg.gz Display(924.00 B)
10mv_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)10mv_validation_2fo-fc_map_coef.cif.gz Display(346.26 KB)
10mv_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)10mv_validation_fo-fc_map_coef.cif.gz Display(345.59 KB)
10mv_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)10mv_validation_2fo-fc_map_coef.mtz Visualize(692.68 KB)
fo-fc (MTZ)10mv_validation_fo-fc_map_coef.mtz Visualize(692.68 KB)

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PDB entries from 2026-04-01

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