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10KZ

N-Alkyl & N-Aryl Aminopyrazole Spirocarbamates: A Two-Pronged Lead Optimization Strategy to Identify Orally Bioavailable Plasma Kallikrein Inhibitors

This is a non-PDB format compatible entry.
Resources
File formatFile name (file size)
PDBx/mmCIF10kz.cif.gz Display(213.94 KB)
10kz.cif
PDBx/mmJSONall10kz.json.gz Display (Tree)(143.24 KB)
10kz.json
no-atom10kz-noatom.json.gz Display (Header)(16.57 KB)
10kz-noatom.json
add only10kz-plus.json.gz Display(882.00 B)
10kz-plus.json
PDBMLall10kz.xml.gz Display(279.62 KB)
10kz.xml
no-atom10kz-noatom.xml.gz Display(27.38 KB)
10kz-noatom.xml
ext-atom10kz-extatom.xml.gz Display(96.70 KB)
10kz-extatom.xml
pdb_nextgenallpdb_000010kz_xyz-enrich.cif.gz Display(222.75 KB)
pdb_000010kz_xyz-enrich.cif
no-atompdb_000010kz_xyz-no-atom-enrich.xml.gz Display(31.10 KB)
pdb_000010kz_xyz-no-atom-enrich.xml
ng-only10kz-plus.json.gz Display(2.32 KB)
10kz-plus.json
RDF10kz.rdf.gz Visualize(79.41 KB)
10kz.rdf
Structure factorsr10kzsf.ent.gz Display(1.21 MB)
r10kzsf.ent
Biological unit (mmCIF format)10kz-assembly1.cif.gz Display(203.57 KB)
10kz-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF10kz_validation.pdf.gz Display(712.92 KB)
10kz_validation.pdf
PDF-full10kz_full_validation.pdf.gz Display(713.35 KB)
10kz_full_validation.pdf
mmCIF10kz_validation.cif.gz Display(22.36 KB)
10kz_validation.cif
XML10kz_validation.xml.gz Display(15.44 KB)
10kz_validation.xml
PNG10kz_multipercentile_validation.png.gz Display(164.03 KB)
10kz_multipercentile_validation.png
SVG10kz_multipercentile_validation.svg.gz Display(958.00 B)
10kz_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)10kz_validation_2fo-fc_map_coef.cif.gz Display(372.93 KB)
10kz_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)10kz_validation_fo-fc_map_coef.cif.gz Display(373.19 KB)
10kz_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)10kz_validation_2fo-fc_map_coef.mtz Visualize(612.76 KB)
fo-fc (MTZ)10kz_validation_fo-fc_map_coef.mtz Visualize(612.76 KB)

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PDB entries from 2026-05-13

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