Summary
| Title: | Selective screening and design to identify inhibitors of Leishmania major pteridine reductase 1. |
| Citation: | Cavazzuti, A.,Paglietti, G.,Hunter, W.N.,Gamarro, F.,Piras, S.,Loriga, M.,Allecca, S.,Corona, P.,McLuskey, K.,Tulloch, L.,Gibellini, F.,Ferrari, S.,Costi, M.P. Discovery of potent pteridine reductase inhibitors to guide antiparasite drug development. Proc.Natl.Acad.Sci.Usa, 105:1448-1453, 2008 PubMed: 18245389DOI: 10.1073/pnas.0704384105 |
| Experimental method: | X-RAY DIFFRACTION (2.4 Å) |
| Deposition date: | 2007-03-22 |
| Release date: | 2007-12-25 |
| Obsoletion date: | 2009-05-05 |
Timeline
Downloads
| File format | File name (file size) | ||
| PDBx/mmCIF | 2p8k.cif.gz Display(433.88 KB) 2p8k.cif | ||
| PDBx/mmJSON | no-atom | 2p8k-noatom.json.gz Display (Header)(22.43 KB) 2p8k-noatom.json | |
| PDBML | all | 2p8k.xml.gz Display(600.93 KB) 2p8k.xml | |
| PDB | pdb2p8k.ent.gz Display(370.52 KB) pdb2p8k.ent | ||
| Structure factors | r2p8ksf.ent.gz Display(856.25 KB) r2p8ksf.ent | ||






