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9MQK

Inactive Kappa-Opioid Receptor with Nb6M, NabFab, and isoquinuclidine compound #020_E1

This is a non-PDB format compatible entry.
Functional Information from GO Data
ChainGOidnamespacecontents
A0004930molecular_functionG protein-coupled receptor activity
A0004985molecular_functionG protein-coupled opioid receptor activity
A0005515molecular_functionprotein binding
A0005654cellular_componentnucleoplasm
A0005739cellular_componentmitochondrion
A0005829cellular_componentcytosol
A0005886cellular_componentplasma membrane
A0006955biological_processimmune response
A0007165biological_processsignal transduction
A0007186biological_processG protein-coupled receptor signaling pathway
A0007193biological_processadenylate cyclase-inhibiting G protein-coupled receptor signaling pathway
A0007200biological_processphospholipase C-activating G protein-coupled receptor signaling pathway
A0007218biological_processneuropeptide signaling pathway
A0007268biological_processchemical synaptic transmission
A0007600biological_processsensory perception
A0007626biological_processlocomotory behavior
A0008528molecular_functionG protein-coupled peptide receptor activity
A0016020cellular_componentmembrane
A0016529cellular_componentsarcoplasmic reticulum
A0019233biological_processsensory perception of pain
A0030315cellular_componentT-tubule
A0030425cellular_componentdendrite
A0030672cellular_componentsynaptic vesicle membrane
A0031635biological_processadenylate cyclase-inhibiting opioid receptor signaling pathway
A0032868biological_processresponse to insulin
A0033603biological_processpositive regulation of dopamine secretion
A0033612molecular_functionreceptor serine/threonine kinase binding
A0033685biological_processnegative regulation of luteinizing hormone secretion
A0035094biological_processresponse to nicotine
A0038003biological_processG protein-coupled opioid receptor signaling pathway
A0038048molecular_functiondynorphin receptor activity
A0042220biological_processresponse to cocaine
A0042383cellular_componentsarcolemma
A0042711biological_processmaternal behavior
A0042734cellular_componentpresynaptic membrane
A0042755biological_processeating behavior
A0042923molecular_functionneuropeptide binding
A0043005cellular_componentneuron projection
A0043025cellular_componentneuronal cell body
A0043204cellular_componentperikaryon
A0043627biological_processresponse to estrogen
A0043679cellular_componentaxon terminus
A0044849biological_processestrous cycle
A0045211cellular_componentpostsynaptic membrane
A0045471biological_processresponse to ethanol
A0046877biological_processregulation of saliva secretion
A0048148biological_processbehavioral response to cocaine
A0050951biological_processsensory perception of temperature stimulus
A0051607biological_processdefense response to virus
A0071222biological_processcellular response to lipopolysaccharide
A0071333biological_processcellular response to glucose stimulus
A1900745biological_processpositive regulation of p38MAPK cascade
A1901381biological_processpositive regulation of potassium ion transmembrane transport
A1903937biological_processresponse to acrylamide
A1904000biological_processpositive regulation of eating behavior
A1990708biological_processconditioned place preference
B0004930molecular_functionG protein-coupled receptor activity
B0004985molecular_functionG protein-coupled opioid receptor activity
B0005515molecular_functionprotein binding
B0005654cellular_componentnucleoplasm
B0005739cellular_componentmitochondrion
B0005829cellular_componentcytosol
B0005886cellular_componentplasma membrane
B0006955biological_processimmune response
B0007165biological_processsignal transduction
B0007186biological_processG protein-coupled receptor signaling pathway
B0007193biological_processadenylate cyclase-inhibiting G protein-coupled receptor signaling pathway
B0007200biological_processphospholipase C-activating G protein-coupled receptor signaling pathway
B0007218biological_processneuropeptide signaling pathway
B0007268biological_processchemical synaptic transmission
B0007600biological_processsensory perception
B0007626biological_processlocomotory behavior
B0008528molecular_functionG protein-coupled peptide receptor activity
B0016020cellular_componentmembrane
B0016529cellular_componentsarcoplasmic reticulum
B0019233biological_processsensory perception of pain
B0030315cellular_componentT-tubule
B0030425cellular_componentdendrite
B0030672cellular_componentsynaptic vesicle membrane
B0031635biological_processadenylate cyclase-inhibiting opioid receptor signaling pathway
B0032868biological_processresponse to insulin
B0033603biological_processpositive regulation of dopamine secretion
B0033612molecular_functionreceptor serine/threonine kinase binding
B0033685biological_processnegative regulation of luteinizing hormone secretion
B0035094biological_processresponse to nicotine
B0038003biological_processG protein-coupled opioid receptor signaling pathway
B0038048molecular_functiondynorphin receptor activity
B0042220biological_processresponse to cocaine
B0042383cellular_componentsarcolemma
B0042711biological_processmaternal behavior
B0042734cellular_componentpresynaptic membrane
B0042755biological_processeating behavior
B0042923molecular_functionneuropeptide binding
B0043005cellular_componentneuron projection
B0043025cellular_componentneuronal cell body
B0043204cellular_componentperikaryon
B0043627biological_processresponse to estrogen
B0043679cellular_componentaxon terminus
B0044849biological_processestrous cycle
B0045211cellular_componentpostsynaptic membrane
B0045471biological_processresponse to ethanol
B0046877biological_processregulation of saliva secretion
B0048148biological_processbehavioral response to cocaine
B0050951biological_processsensory perception of temperature stimulus
B0051607biological_processdefense response to virus
B0071222biological_processcellular response to lipopolysaccharide
B0071333biological_processcellular response to glucose stimulus
B1900745biological_processpositive regulation of p38MAPK cascade
B1901381biological_processpositive regulation of potassium ion transmembrane transport
B1903937biological_processresponse to acrylamide
B1904000biological_processpositive regulation of eating behavior
B1990708biological_processconditioned place preference
Functional Information from PROSITE/UniProt
site_idPS00237
Number of Residues17
DetailsG_PROTEIN_RECEP_F1_1 G-protein coupled receptors family 1 signature. TSIfTLTMMSVDRYIaV
ChainResidueDetails
ATHR144-VAL160

site_idPS00290
Number of Residues7
DetailsIG_MHC Immunoglobulins and major histocompatibility complex proteins signature. YACEVTH
ChainResidueDetails
LTYR192-HIS198
HTYR208-HIS214

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues54
DetailsTransmembrane: {"description":"Helical; Name=1"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues106
DetailsTopological domain: {"description":"Cytoplasmic"}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues46
DetailsTransmembrane: {"description":"Helical; Name=2"}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues74
DetailsTopological domain: {"description":"Extracellular"}
ChainResidueDetails

site_idSWS_FT_FI5
Number of Residues42
DetailsTransmembrane: {"description":"Helical; Name=3"}
ChainResidueDetails

site_idSWS_FT_FI6
Number of Residues44
DetailsTransmembrane: {"description":"Helical; Name=4"}
ChainResidueDetails

site_idSWS_FT_FI7
Number of Residues48
DetailsTransmembrane: {"description":"Helical; Name=5"}
ChainResidueDetails

site_idSWS_FT_FI8
Number of Residues42
DetailsTransmembrane: {"description":"Helical; Name=6"}
ChainResidueDetails

site_idSWS_FT_FI9
Number of Residues42
DetailsTransmembrane: {"description":"Helical; Name=7"}
ChainResidueDetails

site_idSWS_FT_FI10
Number of Residues2
DetailsLipidation: {"description":"S-palmitoyl cysteine","evidences":[{"evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

243083

PDB entries from 2025-10-15

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