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9JDY

Human URAT1 bound with verinurad

This is a non-PDB format compatible entry.
Functional Information from GO Data
ChainGOidnamespacecontents
A0005886cellular_componentplasma membrane
A0006811biological_processmonoatomic ion transport
A0009410biological_processresponse to xenobiotic stimulus
A0015143molecular_functionurate transmembrane transporter activity
A0015711biological_processorganic anion transport
A0015747biological_processurate transport
A0016020cellular_componentmembrane
A0016324cellular_componentapical plasma membrane
A0019725biological_processcellular homeostasis
A0022857molecular_functiontransmembrane transporter activity
A0030165molecular_functionPDZ domain binding
A0031526cellular_componentbrush border membrane
A0032869biological_processcellular response to insulin stimulus
A0046415biological_processurate metabolic process
A0055085biological_processtransmembrane transport
A0070062cellular_componentextracellular exosome
A0097744biological_processrenal urate salt excretion
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues240
DetailsTRANSMEM: Helical => ECO:0000255
ChainResidueDetails
ALEU9-MET29
ASER435-TYR455
AMET466-VAL486
ATRP495-LEU515
APRO146-ALA166
ALEU174-PRO194
AALA195-MET215
ALEU232-ALA252
ALEU260-ALA280
ACYS351-LEU371
AILE378-LEU398
APRO407-PRO427

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphothreonine => ECO:0000250|UniProtKB:Q8CFZ5
ChainResidueDetails
ATHR542

site_idSWS_FT_FI3
Number of Residues2
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255
ChainResidueDetails
AASN56
AASN102

236620

PDB entries from 2025-05-28

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