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9D3C

Gly-,Glu-,(S)-(+)-ketamine bound GluN1a-2B-2D NMDAR

Functional Information from GO Data
ChainGOidnamespacecontents
A0001540molecular_functionamyloid-beta binding
A0004972molecular_functionNMDA glutamate receptor activity
A0005262molecular_functioncalcium channel activity
A0005509molecular_functioncalcium ion binding
A0005515molecular_functionprotein binding
A0005516molecular_functioncalmodulin binding
A0005737cellular_componentcytoplasm
A0005789cellular_componentendoplasmic reticulum membrane
A0005886cellular_componentplasma membrane
A0006811biological_processmonoatomic ion transport
A0006812biological_processmonoatomic cation transport
A0007268biological_processchemical synaptic transmission
A0007420biological_processbrain development
A0008021cellular_componentsynaptic vesicle
A0008542biological_processvisual learning
A0009986cellular_componentcell surface
A0010524biological_processpositive regulation of calcium ion transport into cytosol
A0014069cellular_componentpostsynaptic density
A0015276molecular_functionligand-gated monoatomic ion channel activity
A0015280molecular_functionligand-gated sodium channel activity
A0016020cellular_componentmembrane
A0016594molecular_functionglycine binding
A0016595molecular_functionglutamate binding
A0017146cellular_componentNMDA selective glutamate receptor complex
A0018964biological_processpropylene metabolic process
A0019722biological_processcalcium-mediated signaling
A0022849molecular_functionglutamate-gated calcium ion channel activity
A0030425cellular_componentdendrite
A0034220biological_processmonoatomic ion transmembrane transport
A0034702cellular_componentmonoatomic ion channel complex
A0035235biological_processionotropic glutamate receptor signaling pathway
A0035725biological_processsodium ion transmembrane transport
A0038023molecular_functionsignaling receptor activity
A0042391biological_processregulation of membrane potential
A0043005cellular_componentneuron projection
A0043083cellular_componentsynaptic cleft
A0043195cellular_componentterminal bouton
A0043197cellular_componentdendritic spine
A0044877molecular_functionprotein-containing complex binding
A0045202cellular_componentsynapse
A0045211cellular_componentpostsynaptic membrane
A0045471biological_processresponse to ethanol
A0045944biological_processpositive regulation of transcription by RNA polymerase II
A0046872molecular_functionmetal ion binding
A0048167biological_processregulation of synaptic plasticity
A0048168biological_processregulation of neuronal synaptic plasticity
A0051290biological_processprotein heterotetramerization
A0051968biological_processpositive regulation of synaptic transmission, glutamatergic
A0055074biological_processcalcium ion homeostasis
A0060076cellular_componentexcitatory synapse
A0060079biological_processexcitatory postsynaptic potential
A0070588biological_processcalcium ion transmembrane transport
A0097060cellular_componentsynaptic membrane
A0097553biological_processcalcium ion transmembrane import into cytosol
A0098655biological_processmonoatomic cation transmembrane transport
A0098839cellular_componentpostsynaptic density membrane
A0098878cellular_componentneurotransmitter receptor complex
A0098976biological_processexcitatory chemical synaptic transmission
A0160212molecular_functionglycine-gated cation channel activity
A1903428biological_processpositive regulation of reactive oxygen species biosynthetic process
A1904062biological_processregulation of monoatomic cation transmembrane transport
A1904646biological_processcellular response to amyloid-beta
A1905429biological_processresponse to glycine
A2000463biological_processpositive regulation of excitatory postsynaptic potential
C0001540molecular_functionamyloid-beta binding
C0004972molecular_functionNMDA glutamate receptor activity
C0005262molecular_functioncalcium channel activity
C0005509molecular_functioncalcium ion binding
C0005515molecular_functionprotein binding
C0005516molecular_functioncalmodulin binding
C0005737cellular_componentcytoplasm
C0005789cellular_componentendoplasmic reticulum membrane
C0005886cellular_componentplasma membrane
C0006811biological_processmonoatomic ion transport
C0006812biological_processmonoatomic cation transport
C0007268biological_processchemical synaptic transmission
C0007420biological_processbrain development
C0008021cellular_componentsynaptic vesicle
C0008542biological_processvisual learning
C0009986cellular_componentcell surface
C0010524biological_processpositive regulation of calcium ion transport into cytosol
C0014069cellular_componentpostsynaptic density
C0015276molecular_functionligand-gated monoatomic ion channel activity
C0015280molecular_functionligand-gated sodium channel activity
C0016020cellular_componentmembrane
C0016594molecular_functionglycine binding
C0016595molecular_functionglutamate binding
C0017146cellular_componentNMDA selective glutamate receptor complex
C0018964biological_processpropylene metabolic process
C0019722biological_processcalcium-mediated signaling
C0022849molecular_functionglutamate-gated calcium ion channel activity
C0030425cellular_componentdendrite
C0034220biological_processmonoatomic ion transmembrane transport
C0034702cellular_componentmonoatomic ion channel complex
C0035235biological_processionotropic glutamate receptor signaling pathway
C0035725biological_processsodium ion transmembrane transport
C0038023molecular_functionsignaling receptor activity
C0042391biological_processregulation of membrane potential
C0043005cellular_componentneuron projection
C0043083cellular_componentsynaptic cleft
C0043195cellular_componentterminal bouton
C0043197cellular_componentdendritic spine
C0044877molecular_functionprotein-containing complex binding
C0045202cellular_componentsynapse
C0045211cellular_componentpostsynaptic membrane
C0045471biological_processresponse to ethanol
C0045944biological_processpositive regulation of transcription by RNA polymerase II
C0046872molecular_functionmetal ion binding
C0048167biological_processregulation of synaptic plasticity
C0048168biological_processregulation of neuronal synaptic plasticity
C0051290biological_processprotein heterotetramerization
C0051968biological_processpositive regulation of synaptic transmission, glutamatergic
C0055074biological_processcalcium ion homeostasis
C0060076cellular_componentexcitatory synapse
C0060079biological_processexcitatory postsynaptic potential
C0070588biological_processcalcium ion transmembrane transport
C0097060cellular_componentsynaptic membrane
C0097553biological_processcalcium ion transmembrane import into cytosol
C0098655biological_processmonoatomic cation transmembrane transport
C0098839cellular_componentpostsynaptic density membrane
C0098878cellular_componentneurotransmitter receptor complex
C0098976biological_processexcitatory chemical synaptic transmission
C0160212molecular_functionglycine-gated cation channel activity
C1903428biological_processpositive regulation of reactive oxygen species biosynthetic process
C1904062biological_processregulation of monoatomic cation transmembrane transport
C1904646biological_processcellular response to amyloid-beta
C1905429biological_processresponse to glycine
C2000463biological_processpositive regulation of excitatory postsynaptic potential
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues722
DetailsTOPO_DOM: Extracellular => ECO:0000305|PubMed:36959261
ChainResidueDetails
DPHE28-SER582
DALA675-ASP843
AASN812-ILE835
CSER560-LEU580
CSER628-THR648
CASN812-ILE835

site_idSWS_FT_FI2
Number of Residues64
DetailsTRANSMEM: Helical => ECO:0000269|PubMed:36959261
ChainResidueDetails
DPRO583-PHE604
DTHR654-THR674
DASN844-HIS867
CASN616-PHE627

site_idSWS_FT_FI3
Number of Residues35
DetailsTOPO_DOM: Cytoplasmic => ECO:0000305|PubMed:36959261
ChainResidueDetails
DGLU605-ILE629
DASN642-THR653

site_idSWS_FT_FI4
Number of Residues11
DetailsINTRAMEM: Discontinuously helical => ECO:0000269|PubMed:36959261
ChainResidueDetails
DGLY630-PHE641
CALA649-GLU811

site_idSWS_FT_FI5
Number of Residues2
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:Q62645
ChainResidueDetails
DSER539
DTHR718
BTHR514
BARG519
BSER690
BASP732

site_idSWS_FT_FI6
Number of Residues4
DetailsBINDING: BINDING => ECO:0000269|PubMed:36959261, ECO:0007744|PDB:7YFR
ChainResidueDetails
DTHR541
DARG546
DSER717
DASP759

site_idSWS_FT_FI7
Number of Residues1
DetailsSITE: Functional determinant of NMDA receptors => ECO:0000250
ChainResidueDetails
DASN642
CARG523

site_idSWS_FT_FI8
Number of Residues6
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255
ChainResidueDetails
DASN92
DASN352
DASN366
DASN384
DASN467
DASN569

site_idSWS_FT_FI9
Number of Residues3
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255
ChainResidueDetails
BASN348
BASN444
BASN491

site_idSWS_FT_FI10
Number of Residues2
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000269|PubMed:34321660, ECO:0007744|PDB:7EU8
ChainResidueDetails
BASN542
BASN688

site_idSWS_FT_FI11
Number of Residues2
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255, ECO:0000269|PubMed:36309015, ECO:0000312|PDB:8E93, ECO:0000312|PDB:8E97
ChainResidueDetails
AASN239
CASN239

site_idSWS_FT_FI12
Number of Residues2
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255, ECO:0000269|PubMed:34186027, ECO:0000269|PubMed:36309015, ECO:0000312|PDB:8E92, ECO:0000312|PDB:8E93, ECO:0000312|PDB:8E94, ECO:0000312|PDB:8E96, ECO:0000312|PDB:8E97, ECO:0007744|PDB:7EOQ
ChainResidueDetails
AASN276
CASN276

site_idSWS_FT_FI13
Number of Residues8
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255
ChainResidueDetails
AASN300
AASN440
AASN491
AASN674
CASN300
CASN440
CASN491
CASN674

site_idSWS_FT_FI14
Number of Residues2
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255, ECO:0000269|PubMed:36309015, ECO:0000312|PDB:8E93, ECO:0000312|PDB:8E94, ECO:0000312|PDB:8E96, ECO:0000312|PDB:8E97
ChainResidueDetails
AASN350
CASN350

site_idSWS_FT_FI15
Number of Residues2
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255, ECO:0000269|PubMed:36309015, ECO:0000312|PDB:8E92, ECO:0000312|PDB:8E94, ECO:0000312|PDB:8E97
ChainResidueDetails
AASN368
CASN368

site_idSWS_FT_FI16
Number of Residues2
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255, ECO:0000269|PubMed:34186027, ECO:0000269|PubMed:36309015, ECO:0000269|PubMed:36959261, ECO:0000312|PDB:8E93, ECO:0000312|PDB:8E94, ECO:0000312|PDB:8E97, ECO:0000312|PDB:8E98, ECO:0007744|PDB:7EOQ, ECO:0007744|PDB:7YFR
ChainResidueDetails
AASN471
CASN471

site_idSWS_FT_FI17
Number of Residues2
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255, ECO:0000269|PubMed:34186027, ECO:0000269|PubMed:36309015, ECO:0000312|PDB:8E92, ECO:0000312|PDB:8E93, ECO:0000312|PDB:8E94, ECO:0000312|PDB:8E96, ECO:0000312|PDB:8E97, ECO:0000312|PDB:8E98, ECO:0000312|PDB:8E99, ECO:0007744|PDB:7EOQ
ChainResidueDetails
AASN771
CASN771

237735

PDB entries from 2025-06-18

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