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9CX7

Native human GABAA receptor of beta3-alpha1-gamma2-beta3-alpha2 assembly

Functional Information from GO Data
ChainGOidnamespacecontents
A0004888molecular_functiontransmembrane signaling receptor activity
A0004890molecular_functionGABA-A receptor activity
A0005216molecular_functionmonoatomic ion channel activity
A0005230molecular_functionextracellular ligand-gated monoatomic ion channel activity
A0005254molecular_functionchloride channel activity
A0005886cellular_componentplasma membrane
A0006811biological_processmonoatomic ion transport
A0006821biological_processchloride transport
A0007165biological_processsignal transduction
A0007214biological_processgamma-aminobutyric acid signaling pathway
A0007268biological_processchemical synaptic transmission
A0007399biological_processnervous system development
A0007420biological_processbrain development
A0007612biological_processlearning
A0007613biological_processmemory
A0009410biological_processresponse to xenobiotic stimulus
A0009986cellular_componentcell surface
A0016020cellular_componentmembrane
A0019098biological_processreproductive behavior
A0021549biological_processcerebellum development
A0022851molecular_functionGABA-gated chloride ion channel activity
A0030659cellular_componentcytoplasmic vesicle membrane
A0031410cellular_componentcytoplasmic vesicle
A0034220biological_processmonoatomic ion transmembrane transport
A0034707cellular_componentchloride channel complex
A0035176biological_processsocial behavior
A0035640biological_processexploration behavior
A0042747biological_processcircadian sleep/wake cycle, REM sleep
A0042802molecular_functionidentical protein binding
A0043197cellular_componentdendritic spine
A0045202cellular_componentsynapse
A0045211cellular_componentpostsynaptic membrane
A0048666biological_processneuron development
A0051932biological_processsynaptic transmission, GABAergic
A0060021biological_processroof of mouth development
A0060022biological_processhard palate development
A0060080biological_processinhibitory postsynaptic potential
A0060119biological_processinner ear receptor cell development
A0060384biological_processinnervation
A0061744biological_processmotor behavior
A0071294biological_processcellular response to zinc ion
A0071420biological_processcellular response to histamine
A0072347biological_processresponse to anesthetic
A0090102biological_processcochlea development
A0098982cellular_componentGABA-ergic synapse
A0099634cellular_componentpostsynaptic specialization membrane
A1902476biological_processchloride transmembrane transport
A1902711cellular_componentGABA-A receptor complex
A1904315molecular_functiontransmitter-gated monoatomic ion channel activity involved in regulation of postsynaptic membrane potential
A1904862biological_processinhibitory synapse assembly
B0004888molecular_functiontransmembrane signaling receptor activity
B0004890molecular_functionGABA-A receptor activity
B0005216molecular_functionmonoatomic ion channel activity
B0005230molecular_functionextracellular ligand-gated monoatomic ion channel activity
B0005254molecular_functionchloride channel activity
B0005886cellular_componentplasma membrane
B0006811biological_processmonoatomic ion transport
B0006821biological_processchloride transport
B0007214biological_processgamma-aminobutyric acid signaling pathway
B0008503molecular_functionbenzodiazepine receptor activity
B0016020cellular_componentmembrane
B0016917molecular_functionGABA receptor activity
B0022851molecular_functionGABA-gated chloride ion channel activity
B0030659cellular_componentcytoplasmic vesicle membrane
B0031410cellular_componentcytoplasmic vesicle
B0032590cellular_componentdendrite membrane
B0034220biological_processmonoatomic ion transmembrane transport
B0034707cellular_componentchloride channel complex
B0038023molecular_functionsignaling receptor activity
B0043197cellular_componentdendritic spine
B0045202cellular_componentsynapse
B0045211cellular_componentpostsynaptic membrane
B0051932biological_processsynaptic transmission, GABAergic
B0060078biological_processregulation of postsynaptic membrane potential
B0098794cellular_componentpostsynapse
B0098982cellular_componentGABA-ergic synapse
B0099634cellular_componentpostsynaptic specialization membrane
B1902476biological_processchloride transmembrane transport
B1902710cellular_componentGABA receptor complex
B1902711cellular_componentGABA-A receptor complex
B1904315molecular_functiontransmitter-gated monoatomic ion channel activity involved in regulation of postsynaptic membrane potential
B1904862biological_processinhibitory synapse assembly
C0004888molecular_functiontransmembrane signaling receptor activity
C0004890molecular_functionGABA-A receptor activity
C0005216molecular_functionmonoatomic ion channel activity
C0005230molecular_functionextracellular ligand-gated monoatomic ion channel activity
C0005254molecular_functionchloride channel activity
C0005515molecular_functionprotein binding
C0005886cellular_componentplasma membrane
C0006811biological_processmonoatomic ion transport
C0006821biological_processchloride transport
C0007214biological_processgamma-aminobutyric acid signaling pathway
C0007268biological_processchemical synaptic transmission
C0008503molecular_functionbenzodiazepine receptor activity
C0009791biological_processpost-embryonic development
C0016020cellular_componentmembrane
C0022851molecular_functionGABA-gated chloride ion channel activity
C0030424cellular_componentaxon
C0030425cellular_componentdendrite
C0030534biological_processadult behavior
C0030659cellular_componentcytoplasmic vesicle membrane
C0031410cellular_componentcytoplasmic vesicle
C0032590cellular_componentdendrite membrane
C0034220biological_processmonoatomic ion transmembrane transport
C0034707cellular_componentchloride channel complex
C0042995cellular_componentcell projection
C0045202cellular_componentsynapse
C0045211cellular_componentpostsynaptic membrane
C0051932biological_processsynaptic transmission, GABAergic
C0060078biological_processregulation of postsynaptic membrane potential
C0071420biological_processcellular response to histamine
C0098794cellular_componentpostsynapse
C0098982cellular_componentGABA-ergic synapse
C0099634cellular_componentpostsynaptic specialization membrane
C1902476biological_processchloride transmembrane transport
C1902711cellular_componentGABA-A receptor complex
C1904315molecular_functiontransmitter-gated monoatomic ion channel activity involved in regulation of postsynaptic membrane potential
C1904862biological_processinhibitory synapse assembly
D0004888molecular_functiontransmembrane signaling receptor activity
D0004890molecular_functionGABA-A receptor activity
D0005216molecular_functionmonoatomic ion channel activity
D0005230molecular_functionextracellular ligand-gated monoatomic ion channel activity
D0005254molecular_functionchloride channel activity
D0005886cellular_componentplasma membrane
D0006811biological_processmonoatomic ion transport
D0006821biological_processchloride transport
D0007165biological_processsignal transduction
D0007214biological_processgamma-aminobutyric acid signaling pathway
D0007268biological_processchemical synaptic transmission
D0007399biological_processnervous system development
D0007420biological_processbrain development
D0007612biological_processlearning
D0007613biological_processmemory
D0009410biological_processresponse to xenobiotic stimulus
D0009986cellular_componentcell surface
D0016020cellular_componentmembrane
D0019098biological_processreproductive behavior
D0021549biological_processcerebellum development
D0022851molecular_functionGABA-gated chloride ion channel activity
D0030659cellular_componentcytoplasmic vesicle membrane
D0031410cellular_componentcytoplasmic vesicle
D0034220biological_processmonoatomic ion transmembrane transport
D0034707cellular_componentchloride channel complex
D0035176biological_processsocial behavior
D0035640biological_processexploration behavior
D0042747biological_processcircadian sleep/wake cycle, REM sleep
D0042802molecular_functionidentical protein binding
D0043197cellular_componentdendritic spine
D0045202cellular_componentsynapse
D0045211cellular_componentpostsynaptic membrane
D0048666biological_processneuron development
D0051932biological_processsynaptic transmission, GABAergic
D0060021biological_processroof of mouth development
D0060022biological_processhard palate development
D0060080biological_processinhibitory postsynaptic potential
D0060119biological_processinner ear receptor cell development
D0060384biological_processinnervation
D0061744biological_processmotor behavior
D0071294biological_processcellular response to zinc ion
D0071420biological_processcellular response to histamine
D0072347biological_processresponse to anesthetic
D0090102biological_processcochlea development
D0098982cellular_componentGABA-ergic synapse
D0099634cellular_componentpostsynaptic specialization membrane
D1902476biological_processchloride transmembrane transport
D1902711cellular_componentGABA-A receptor complex
D1904315molecular_functiontransmitter-gated monoatomic ion channel activity involved in regulation of postsynaptic membrane potential
D1904862biological_processinhibitory synapse assembly
E0004888molecular_functiontransmembrane signaling receptor activity
E0004890molecular_functionGABA-A receptor activity
E0005216molecular_functionmonoatomic ion channel activity
E0005230molecular_functionextracellular ligand-gated monoatomic ion channel activity
E0005254molecular_functionchloride channel activity
E0005515molecular_functionprotein binding
E0005886cellular_componentplasma membrane
E0006811biological_processmonoatomic ion transport
E0006821biological_processchloride transport
E0007214biological_processgamma-aminobutyric acid signaling pathway
E0008503molecular_functionbenzodiazepine receptor activity
E0016020cellular_componentmembrane
E0022851molecular_functionGABA-gated chloride ion channel activity
E0030424cellular_componentaxon
E0030425cellular_componentdendrite
E0030659cellular_componentcytoplasmic vesicle membrane
E0030672cellular_componentsynaptic vesicle membrane
E0031410cellular_componentcytoplasmic vesicle
E0032590cellular_componentdendrite membrane
E0034220biological_processmonoatomic ion transmembrane transport
E0034707cellular_componentchloride channel complex
E0038023molecular_functionsignaling receptor activity
E0042995cellular_componentcell projection
E0043025cellular_componentneuronal cell body
E0045202cellular_componentsynapse
E0045211cellular_componentpostsynaptic membrane
E0051932biological_processsynaptic transmission, GABAergic
E0060077cellular_componentinhibitory synapse
E0060078biological_processregulation of postsynaptic membrane potential
E0098794cellular_componentpostsynapse
E0098982cellular_componentGABA-ergic synapse
E0099505biological_processregulation of presynaptic membrane potential
E0099507molecular_functionligand-gated monoatomic ion channel activity involved in regulation of presynaptic membrane potential
E0099634cellular_componentpostsynaptic specialization membrane
E1902476biological_processchloride transmembrane transport
E1902711cellular_componentGABA-A receptor complex
E1904315molecular_functiontransmitter-gated monoatomic ion channel activity involved in regulation of postsynaptic membrane potential
E1904862biological_processinhibitory synapse assembly
Functional Information from PROSITE/UniProt
site_idPS00236
Number of Residues15
DetailsNEUROTR_ION_CHANNEL Neurotransmitter-gated ion-channels signature. CqLqLhnFPmDehsC
ChainResidueDetails
CCYS151-CYS165
ACYS136-CYS150
ECYS138-CYS152
BCYS139-CYS153

site_idPS00290
Number of Residues7
DetailsIG_MHC Immunoglobulins and major histocompatibility complex proteins signature. FSCNVRH
ChainResidueDetails
KPHE430-HIS436
LTYR191-HIS197

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues239
DetailsTOPO_DOM: Extracellular => ECO:0000305
ChainResidueDetails
EASN1-LYS221
EARG273-THR283
EASN414-PRO423
DLEU268-LYS279

site_idSWS_FT_FI2
Number of Residues79
DetailsTRANSMEM: Helical => ECO:0000255
ChainResidueDetails
EILE222-VAL242
EALA253-ALA272
EALA284-ALA304
ESER393-LEU413
DILE222-ILE242
DSER247-HIS267
DALA280-ASN303
DILE423-TYR445

site_idSWS_FT_FI3
Number of Residues96
DetailsTOPO_DOM: Cytoplasmic => ECO:0000305
ChainResidueDetails
ESER243-PRO252
ETHR305-MET392
DASN243-ALA246
DTYR304-ALA422

site_idSWS_FT_FI4
Number of Residues1
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:P14867
ChainResidueDetails
EARG66
CASN90

site_idSWS_FT_FI5
Number of Residues1
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:P62813
ChainResidueDetails
ETHR129
APHE200
DASP95
DPHE200

site_idSWS_FT_FI6
Number of Residues2
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255
ChainResidueDetails
EASN10
EASN110
ATHR202
DTYR97
DSER156
DTHR202

site_idSWS_FT_FI7
Number of Residues1
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255
ChainResidueDetails
BASN11
DGLU155

site_idSWS_FT_FI8
Number of Residues1
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000269|PubMed:29950725, ECO:0000269|PubMed:30602789, ECO:0007744|PDB:6D6T, ECO:0007744|PDB:6D6U, ECO:0007744|PDB:6I53
ChainResidueDetails
BASN111
DTYR157

site_idSWS_FT_FI9
Number of Residues2
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000269|PubMed:24909990, ECO:0000269|PubMed:35355020, ECO:0007744|PDB:7QN7
ChainResidueDetails
AASN8
DASN8

site_idSWS_FT_FI10
Number of Residues2
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000269|PubMed:24909990, ECO:0000269|PubMed:30602789, ECO:0000269|PubMed:35355020, ECO:0007744|PDB:6I53, ECO:0007744|PDB:7QN7
ChainResidueDetails
AASN80
DASN80

site_idSWS_FT_FI11
Number of Residues2
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000269|PubMed:24909990, ECO:0000269|PubMed:30140029, ECO:0000269|PubMed:30602789, ECO:0000269|PubMed:35355020, ECO:0007744|PDB:6A96, ECO:0007744|PDB:6I53, ECO:0007744|PDB:7QN7
ChainResidueDetails
AASN149
DASN149

236371

PDB entries from 2025-05-21

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