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9BBB

Human CYP3A4 bound to an inhibitor

This is a non-PDB format compatible entry.
Functional Information from PROSITE/UniProt
site_idPS00086
Number of Residues10
DetailsCYTOCHROME_P450 Cytochrome P450 cysteine heme-iron ligand signature. FGsGPRNCIG
ChainResidueDetails
APHE435-GLY444

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues20
DetailsTRANSMEM: Helical => ECO:0000255
ChainResidueDetails
AALA2-THR42

site_idSWS_FT_FI2
Number of Residues1
DetailsBINDING: axial binding residue => ECO:0007744|PDB:1TQN, ECO:0007744|PDB:1W0G
ChainResidueDetails
AASN462

222415

PDB entries from 2024-07-10

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