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8XVJ

Cryo-EM structure of ETAR bound with Macitentan

This is a non-PDB format compatible entry.
Functional Information from PROSITE/UniProt
site_idPS00237
Number of Residues17
DetailsG_PROTEIN_RECEP_F1_1 G-protein coupled receptors family 1 signature. ITVlNLCALSVDRYRaV
ChainResidueDetails
RILE171-VAL187

site_idPS00290
Number of Residues7
DetailsIG_MHC Immunoglobulins and major histocompatibility complex proteins signature. YICNVNH
ChainResidueDetails
HTYR208-HIS214
LTYR194-HIS200

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsACT_SITE: Proton donor => ECO:0000255|PROSITE-ProRule:PRU01100
ChainResidueDetails
RALA-131

site_idSWS_FT_FI2
Number of Residues1
DetailsACT_SITE: Nucleophile => ECO:0000255|PROSITE-ProRule:PRU01100
ChainResidueDetails
RGLU-18

site_idSWS_FT_FI3
Number of Residues21
DetailsTRANSMEM: Helical; Name=1 => ECO:0000255
ChainResidueDetails
RTYR81-LEU102

site_idSWS_FT_FI4
Number of Residues32
DetailsTOPO_DOM: Cytoplasmic => ECO:0000255
ChainResidueDetails
RARG103-ARG112
RASP182-GLU205

site_idSWS_FT_FI5
Number of Residues19
DetailsTRANSMEM: Helical; Name=2 => ECO:0000255
ChainResidueDetails
RASN113-ILE132

site_idSWS_FT_FI6
Number of Residues70
DetailsTOPO_DOM: Extracellular => ECO:0000255
ChainResidueDetails
RASP133-LYS159
RGLU230-ASP256
RLYS329-LEU347

site_idSWS_FT_FI7
Number of Residues21
DetailsTRANSMEM: Helical; Name=3 => ECO:0000255
ChainResidueDetails
RLEU160-VAL181

site_idSWS_FT_FI8
Number of Residues23
DetailsTRANSMEM: Helical; Name=4 => ECO:0000255
ChainResidueDetails
RILE206-PHE229

site_idSWS_FT_FI9
Number of Residues21
DetailsTRANSMEM: Helical; Name=5 => ECO:0000255
ChainResidueDetails
RTRP257-MET278

site_idSWS_FT_FI10
Number of Residues21
DetailsTRANSMEM: Helical; Name=6 => ECO:0000255
ChainResidueDetails
RTHR307-LEU328

site_idSWS_FT_FI11
Number of Residues24
DetailsTRANSMEM: Helical; Name=7 => ECO:0000255
ChainResidueDetails
RLEU348-VAL372

site_idSWS_FT_FI12
Number of Residues1
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255
ChainResidueDetails
RASN62

site_idSWS_FT_FI13
Number of Residues2
DetailsBINDING: axial binding residue
ChainResidueDetails
RTRP1012
RILE1107

224201

PDB entries from 2024-08-28

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