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8VV8

Crystal Structure of EHMT2 bound to EZM8266

This is a non-PDB format compatible entry.
Functional Information from GO Data
ChainGOidnamespacecontents
A0002039molecular_functionp53 binding
A0005634cellular_componentnucleus
A0008270molecular_functionzinc ion binding
A0016279molecular_functionprotein-lysine N-methyltransferase activity
A0042054molecular_functionhistone methyltransferase activity
B0002039molecular_functionp53 binding
B0005634cellular_componentnucleus
B0008270molecular_functionzinc ion binding
B0016279molecular_functionprotein-lysine N-methyltransferase activity
B0042054molecular_functionhistone methyltransferase activity
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues126
DetailsDomain: {"description":"Pre-SET","evidences":[{"source":"PROSITE-ProRule","id":"PRU00157","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues234
DetailsDomain: {"description":"SET","evidences":[{"source":"PROSITE-ProRule","id":"PRU00190","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues32
DetailsDomain: {"description":"Post-SET"}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues44
DetailsRegion: {"description":"Interaction with histone H3","evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI5
Number of Residues32
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"20084102","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"24900801","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"2O8J","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"4NVQ","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI6
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"20084102","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"2O8J","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"4NVQ","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI7
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"27648579","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"5T0M","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI8
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"20084102","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"2O8J","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI9
Number of Residues2
DetailsSite: {"description":"Histone H3K9me binding","evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

249524

PDB entries from 2026-02-18

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