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8VOF

GI targeted CpPI4K inhibitor

This is a non-PDB format compatible entry.
Functional Information from PROSITE/UniProt
site_idPS00675
Number of Residues14
DetailsSIGMA54_INTERACT_1 Sigma-54 interaction domain ATP-binding region A signature. VVLiGDSGVGKsnL
ChainResidueDetails
BVAL14-LEU27

site_idPS00915
Number of Residues15
DetailsPI3_4_KINASE_1 Phosphatidylinositol 3- and 4-kinases signature 1. VKcg.DDLRQEllafQ
ChainResidueDetails
AVAL548-GLN562

site_idPS00916
Number of Residues21
DetailsPI3_4_KINASE_2 Phosphatidylinositol 3- and 4-kinases signature 2. ScAgycLvcYLLqVkDRHngN
ChainResidueDetails
ASER641-ASN661

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBINDING: BINDING => ECO:0000269|PubMed:16905101, ECO:0000269|PubMed:17007872, ECO:0000269|PubMed:17030804, ECO:0007744|PDB:2D7C, ECO:0007744|PDB:2GZD, ECO:0007744|PDB:2GZH, ECO:0007744|PDB:2HV8, ECO:0007744|PDB:5EZ5
ChainResidueDetails
BGLY18
BASN124
BSER154

site_idSWS_FT_FI2
Number of Residues1
DetailsBINDING: BINDING => ECO:0007744|PDB:2D7C, ECO:0007744|PDB:2GZD, ECO:0007744|PDB:2GZH, ECO:0007744|PDB:2HV8, ECO:0007744|PDB:5EZ5
ChainResidueDetails
BASN37

site_idSWS_FT_FI3
Number of Residues1
DetailsBINDING: BINDING => ECO:0000269|PubMed:16905101, ECO:0000269|PubMed:17007872, ECO:0000269|PubMed:17030804, ECO:0007744|PDB:1OIW, ECO:0007744|PDB:4D0L, ECO:0007744|PDB:4D0M, ECO:0007744|PDB:5C46, ECO:0007744|PDB:5FBL
ChainResidueDetails
BASP66

site_idSWS_FT_FI4
Number of Residues1
DetailsMOD_RES: N-acetylglycine => ECO:0000269|Ref.11
ChainResidueDetails
BGLY2
AARG323

site_idSWS_FT_FI5
Number of Residues1
DetailsMOD_RES: Cysteine methyl ester => ECO:0000255
ChainResidueDetails
BCYS213

site_idSWS_FT_FI6
Number of Residues2
DetailsLIPID: S-geranylgeranyl cysteine => ECO:0000269|PubMed:24023390
ChainResidueDetails
BCYS212
BCYS213

site_idSWS_FT_FI7
Number of Residues1
DetailsCARBOHYD: (Microbial infection) N-beta-linked (GlcNAc) arginine => ECO:0000269|PubMed:32974215
ChainResidueDetails
BARG4

224572

PDB entries from 2024-09-04

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